⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| Hydrochloric Acid SCHEMBL29689430 | 0.98 | — | — | |
| Phenol SCHEMBL29688819 | 0.85 | CA12 (0.34) | — | |
| SCHEMBL436647 | 0.81 | CHRNB2 (0.33) | — | |
| SCHEMBL3810433 | 0.81 | HTR2C (0.40) | — | |
| SCHEMBL1300630 | 0.78 | — | — | |
| SCHEMBL30579615 | 0.68 | HTR2C (0.34) | — | |
| SCHEMBL860227 | 0.67 | HRH1 (0.41) | — | |
| SCHEMBL1000578 | 0.67 | — | — | |
| SCHEMBL1174158 | 0.65 | — | — | |
| SCHEMBL368150 | 0.65 | MAPT (0.37) | — |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 234 patents. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| CN-118745244-A | Method for preparing polycarbonate by proton type ionic liquid catalysis | 中国科学院过程工程研究所 | 2024-10-08 | — | — | CN | claimed |
| EP-3512905-B1 | METHOD FOR PRODUCING A POLYBENZAZOL POLYMER (P) | BASF SE (DE) | 2022-08-24 | — | — | EP | claimed |
| US-20200407508-A1 | METHOD FOR PRODUCING FIBERS, FILMS AND MOLDINGS OF A POLYBENZAZOLE POLYMER (P) | BASF SE (DE) | 2020-12-31 | — | — | US | claimed |
| EP-1812382-B1 | METHOD FOR PRODUCING POLYISOCYANATES | BASF SE (DE) | 2013-01-23 | — | — | EP | claimed |
| EP-2130827-B1 | METHOD FOR PRODUCING QUINOLONE CARBOXYLIC ACID DERIVATIVE | DAIICHI SANKYO CO LTD (JP) | 2012-02-01 | — | — | EP | claimed |
| EP-1711472-B1 | MEHTOD FOR PRODUCING IONIC LIQUIDS | BASF SE (DE) | 2011-05-25 | — | — | EP | claimed |
| US-7875722-B2 | having high antibacterial activity and high safety, at high yield and in a simple manner; one-pot process | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2011-01-25 | — | — | US | claimed |
| US-20090112017-A1 | METHOD FOR PRODUCING POLYISOCYANATES | BASF AKTIENGESSELLSCHAFT (DE) | 2009-04-30 | — | — | US | claimed |
| EP-1644395-B1 | PROCESSES FOR PREPARING 4'AZIDO NUCLEOSIDE DERIVATIVES | HOFFMANN LA ROCHE (CH) | 2006-11-22 | — | — | EP | claimed |
| US-7087778-B2 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. (JP) | 2006-08-08 | — | — | US | claimed |
| WO-2005118527-A2 | FLUOROUS CAPPING REAGENTS, AND METHODS FOR PEPTIDE PURIFICATION | TRUSTEES OF TUFTS COLLEGE (US) | 2005-12-15 | — | — | WO | claimed |
| US-20050027119-A1 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. | 2005-02-03 | — | — | US | claimed |
| EP-1363890-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | Millennium Pharmaceuticals, Inc. (US) | 2003-11-26 | — | — | EP | claimed |
| WO-2002062766-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | MILLENNIUM PHARMACEUTICALS, INC. (US) | 2002-08-15 | — | — | WO | claimed |
| EP-1211254-A1 | PROCESS FOR THE PREPARATION OF BENZOXAZINE DERIVATIVES AND INTERMEDIATES THEREFOR | DAIICHI PHARMACEUTICAL CO., LTD. (JP) | 2002-06-05 | — | — | EP | claimed |
| EP-1204645-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | Millennium Pharmaceuticals, Inc. (US) | 2002-05-15 | — | — | EP | claimed |
| WO-2001010842-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | MILLENNIUM PHARMACEUTICALS, INC. (US) | 2001-02-15 | — | — | WO | claimed |
| US-4889911-A | ESTERIFICATION, ESTER INTERCHANGE; CATALYSIS WITH HETEROCYCLIC NITROGEN COMPOUND | BAYER AKTIENGESELLSCHAFT (DE) | 1989-12-26 | — | — | US | claimed |
| EP-0303931-A2 | Process for the fabrication of thermotropic, wholly aromatic polyesters and polyestercarbonates | BAYER AG (DE) | 1989-02-22 | — | — | EP | claimed |
| US-12630744-B2 | Polishing compositions and methods of use thereof | FUJIFILM ELECTRONIC MATERIALS U.S.A., INC. (US) | 2026-05-19 | — | — | US | disclosed |
| EP-4688987-A1 | POLISHING COMPOSITIONS AND METHODS OF USE THEREOF | FUJIFILM Electronic Materials U.S.A, Inc. (US) | 2026-02-11 | — | — | EP | disclosed |
| US-20260015438-A1 | Photopolymerizable Compositions Including a Polyurethane Methacrylate Polymer Prepared Using a Polycarbonate Diol, Articles, and Methods | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2026-01-15 | — | — | US | disclosed |
| EP-3917445-B1 | METHODS OF MAKING AND POSTPROCESSING ORTHODONTIC ARTICLES | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2025-11-05 | — | — | EP | disclosed |
| US-12440560-B2 | Substituted pyrimidines as vaccine adjuvants | Sumitomo Pharma Co., Ltd. (JP) | 2025-10-14 | — | — | US | disclosed |
| EP-3603619-B1 | VACCINE ADJUVANT FORMULATION | SUMITOMO PHARMA CO LTD (JP) | 2025-08-13 | — | — | EP | disclosed |
| US-12351668-B2 | Orthodontic articles comprising polymerized composition with pendent cyclic moieties, methods, and polymerizable compositions | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2025-07-08 | — | — | US | disclosed |
| EP-3973007-B1 | ORTHODONTIC ARTICLES COMPRISING POLYMERIZED COMPOSITION WITH PENDENT CYCLIC MOIETIES, METHODS, AND POLYMERIZABLE COMPOSITIONS | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2025-06-25 | — | — | EP | disclosed |
| US-12297316-B2 | Orthodontic articles prepared using a polycarbonate diol, polymerizable compositions, and methods of making the articles | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2025-05-13 | — | — | US | disclosed |
| CN-119219534-B | Synthesis method and application of o-amino disulfide and benazolin ethyl ester key intermediate 4-chlorobenzothiazole | 鄂尔多斯应用技术学院 | 2025-04-08 | — | — | CN | disclosed |
| WO-2025057020-A1 | PHOTOPOLYMERIZABLE COMPOSITIONS INCLUDING UREA/ACRYLAMIDE FUNCTIONAL COMPONENT, ARTICLES AND METHODS | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2025-03-20 | — | — | WO | disclosed |
| US-20250009479-A1 | Orthodontic Articles and Methods of Making and Postprocessing Same | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2025-01-09 | — | — | US | disclosed |
| CN-119219534-A | Synthesis method and application of o-amino disulfide and benazolin ethyl ester key intermediate 4-chlorobenzothiazole | 鄂尔多斯应用技术学院 | 2024-12-31 | — | — | CN | disclosed |
| US-12121413-B2 | Orthodontic articles and methods of making and postprocessing same | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY (US) | 2024-10-22 | — | — | US | disclosed |
| US-20240327675-A1 | POLISHING COMPOSITIONS AND METHODS OF USE THEREOF | FUJIFILM ELECTRONIC MATERIALS U.S.A., INC. | 2024-10-03 | — | — | US | disclosed |
| WO-2024206301-A1 | POLISHING COMPOSITIONS AND METHODS OF USE THEREOF | FUJIFILM ELECTRONIC MATERIALS U.S.A., INC. (US) | 2024-10-03 | — | — | WO | disclosed |
| CN-110650729-B | Vaccine adjuvant formulations | 住友制药株式会社 | 2024-08-20 | — | — | CN | disclosed |
| US-20240270893-A1 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, POLYMERIZABLE COMPOSITIONS, AND METHODS OF MAKING THE ARTICLES | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2024-08-15 | — | — | US | disclosed |
| US-20240245766-A1 | PYRIMIDINE COMPOUND | Sumitomo Pharma Co., Ltd. (JP) | 2024-07-25 | — | — | US | disclosed |
| WO-2024118398-A1 | POLISHING COMPOSITIONS AND METHODS OF USE THEREOF | FUJIFILM ELECTRONIC MATERIALS U.S.A., INC. (US) | 2024-06-06 | — | — | WO | disclosed |
| US-20240174892-A1 | POLISHING COMPOSITIONS AND METHODS OF USE THEREOF | FUJIFILM ELECTRONIC MATERIALS U.S.A., INC. | 2024-05-30 | — | — | US | disclosed |
| US-11945900-B2 | Orthodontic articles prepared using a polycarbonate diol, polymerizable compositions, and methods of making the articles | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2024-04-02 | — | — | US | disclosed |
| US-11911466-B2 | Substituted pyrimidines as vaccine adjuvants | Sumitomo Pharma Co., Ltd. (JP) | 2024-02-27 | — | — | US | disclosed |
| US-11833247-B2 | Vaccine adjuvant formulation | Sumitomo Pharma Co., Ltd. (JP) | 2023-12-05 | — | — | US | disclosed |
| US-20230322966-A1 | Photopolymerizable Compositions Including a Polyurethane Methacrylate Polymer Prepared Using a Polycarbonate Diol, Articles, and Methods | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2023-10-12 | — | — | US | disclosed |
| US-11771086-B2 | Pest control composition including novel iminopyridine derivative | MMAG CO., LTD. (JP) | 2023-10-03 | — | — | US | disclosed |
| EP-3868741-B1 | COMPOSITION COMPRISING A PYRIMIDINE COMPOUND AND A PATHOGEN DERIVED ANTIGEN | SUMITOMO PHARMA CO LTD (JP) | 2023-08-30 | — | — | EP | disclosed |
| US-11708428-B2 | Photopolymerizable compositions including a polyurethane methacrylate polymer prepared using a polycarbonate diol, articles, and methods | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2023-07-25 | — | — | US | disclosed |
| US-11584874-B2 | Increased saturation of ice melting compositions and methods of use | BASF SE (DE) | 2023-02-21 | — | — | US | disclosed |
| US-20220273563-A1 | VACCINE ADJUVANT FORMULATION | Sumitomo Pharma Co., Ltd. (JP) | 2022-09-01 | — | — | US | disclosed |
| EP-3512905-B1 | METHOD FOR PRODUCING A POLYBENZAZOL POLYMER (P) | BASF SE (DE) | 2022-08-24 | — | — | EP | disclosed |
| US-20220242991-A1 | Orthodontic Articles Comprising Polymerized Composition with Pendent Cyclic Moieties, Methods, and Polymerizable Compositions | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2022-08-04 | — | — | US | disclosed |
| US-20220226468-A1 | PYRIMIDINE COMPOUND | Sumitomo Pharma Co., Ltd. (JP) | 2022-07-21 | — | — | US | disclosed |
| CN-111771885-B | Pest control composition comprising novel iminopyridine derivatives | 株式会社MMAG | 2022-05-17 | — | — | CN | disclosed |
| CN-112244015-B | Pest control composition comprising novel iminopyridine derivatives | 株式会社MMAG | 2022-05-17 | — | — | CN | disclosed |
| EP-3973007-A1 | ORTHODONTIC ARTICLES COMPRISING POLYMERIZED COMPOSITION WITH PENDENT CYCLIC MOIETIES, METHODS, AND POLYMERIZABLE COMPOSITIONS | 3M Innovative Properties Company (US) | 2022-03-30 | — | — | EP | disclosed |
| US-20220056258-A1 | ORTHODONTIC ARTICLES COMPRISING POLYESTER URETHANE (METH)ACRYLATE POLYMER AND MONOFUNCTIONAL (METH)ACRYLATE MONOMER, METHODS, AND POLYMERIZABLE COMPOSITIONS | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2022-02-24 | — | — | US | disclosed |
| US-11253476-B2 | Vaccine adjuvant formulation | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2022-02-22 | — | — | US | disclosed |
| US-20220023007-A1 | Orthodontic Articles and Methods of Making and Postprocessing Same | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2022-01-27 | — | — | US | disclosed |
| US-11225535-B2 | Photopolymerizable compositions including a polyurethane methacrylate polymer prepared using a polycarbonate diol, articles, and methods | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2022-01-18 | — | — | US | disclosed |
| EP-3917445-A1 | ORTHODONTIC ARTICLES AND METHODS OF MAKING AND POSTPROCESSING SAME | 3M Innovative Properties Company (US) | 2021-12-08 | — | — | EP | disclosed |
| CN-112118802-B | Orthodontic articles prepared using polycarbonate diols and methods of making the same | 3M创新有限公司 | 2021-12-07 | — | — | CN | disclosed |
| CN-113767131-A | Orthodontic articles, methods, and polymerizable compositions comprising polymeric compositions having pendant ring moieties | 3M创新有限公司 | 2021-12-07 | — | — | CN | disclosed |
| US-20210361389-A1 | HYDRATED ORTHODONTIC ARTICLES, KITS, AND METHODS OF MAKING SAME | 3M INNOVATIVE PROPERTIES COMPANY | 2021-11-25 | — | — | US | disclosed |
| US-20210355262-A1 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, AND METHODS OF MAKING SAME | 3M INNOVATIVE PROPERTIES COMPANY | 2021-11-18 | — | — | US | disclosed |
| US-20210301042-A1 | PHOTOPOLYMERIZABLE COMPOSITIONS INCLUDING A POLYURETHANE METHACRYLATE POLYMER PREPARED USING A POLYCARBONATE DIOL, ARTICLES, AND METHODS | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2021-09-30 | — | — | US | disclosed |
| EP-3883521-A1 | ORTHODONTIC ARTICLES COMPRISING POLYESTER URETHANE (METH)ACRYLATE POLYMER AND MONOFUNCTIONAL (METH)ACRYLATE MONOMER, METHODS, AND POLYMERIZABLE COMPOSITIONS | 3M Innovative Properties Company (US) | 2021-09-29 | — | — | EP | disclosed |
| CN-113286560-A | Orthodontic articles and methods of making and post-treating the same | 3M创新有限公司 | 2021-08-20 | — | — | CN | disclosed |
| CN-113015511-A | Orthodontic articles, methods, and polymerizable compositions comprising polyester urethane (meth) acrylate polymers and monofunctional (meth) acrylate monomers | 3M创新有限公司 | 2021-06-22 | — | — | CN | disclosed |
| US-20210171701-A1 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, POLYMERIZABLE COMPOSITIONS, AND METHODS OF MAKING THE ARTICLES | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2021-06-10 | — | — | US | disclosed |
| US-20210163664-A1 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, AND METHODS OF MAKING SAME | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2021-06-03 | — | — | US | disclosed |
| EP-3813764-A2 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, POLYMERIZABLE COMPOSITIONS, AND METHODS OF MAKING THE ARTICLES | 3M Innovative Properties Company (US) | 2021-05-05 | — | — | EP | disclosed |
| EP-3360864-B1 | PYRIMIDINE COMPOUND | SUMITOMO DAINIPPON PHARMA CO LTD (JP) | 2021-04-28 | — | — | EP | disclosed |
| EP-3806774-A1 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, AND METHODS OF MAKING SAME | 3M Innovative Properties Company (US) | 2021-04-21 | — | — | EP | disclosed |
| US-20210095056-A1 | PHOTOPOLYMERIZABLE COMPOSITIONS INCLUDING A POLYURETHANE METHACRYLATE POLYMER PREPARED USING A POLYCARBONATE DIOL, ARTICLES, AND METHODS | SOLVENTUM INTELLECTUAL PROPERTIES COMPANY | 2021-04-01 | — | — | US | disclosed |
| WO-2021037349-A1 | MULTI-COMPONENT CROSSLINKABLE MATERIALS BASED ON ORGANYLOXYSILANE-TERMINATED POLYMERS AND EPOXY-FUNCTIONAL COMPOUNDS | WACKER CHEMIE AG (DE) | 2021-03-04 | — | — | WO | disclosed |
| CN-112384188-A | Orthodontic articles made using polycarbonate diols, polymerizable compositions, and methods of making articles | 3M创新有限公司 | 2021-02-19 | — | — | CN | disclosed |
| US-20210008197-A1 | PYRIMIDINE COMPOUND | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2021-01-14 | — | — | US | disclosed |
| US-20200407508-A1 | METHOD FOR PRODUCING FIBERS, FILMS AND MOLDINGS OF A POLYBENZAZOLE POLYMER (P) | BASF SE (DE) | 2020-12-31 | — | — | US | disclosed |
| EP-3752123-A1 | PHOTOPOLYMERIZABLE COMPOSITIONS INCLUDING A POLYURETHANE METHACRYLATE POLYMER PREPARED USING A POLYCARBONATE DIOL, ARTICLES, AND METHODS | 3M Innovative Properties Company (US) | 2020-12-23 | — | — | EP | disclosed |
| CN-112118802-A | Orthodontic articles prepared using polycarbonate diols and methods of making the same | 3M创新有限公司 | 2020-12-22 | — | — | CN | disclosed |
| CN-112105332-A | Photopolymerizable compositions, articles, and methods comprising urethane methacrylate polymers prepared using polycarbonate diols | 3M创新有限公司 | 2020-12-18 | — | — | CN | disclosed |
| WO-2020234775-A1 | ORTHODONTIC ARTICLES COMPRISING POLYMERIZED COMPOSITION WITH PENDENT CYCLIC MOIETIES, METHODS, AND POLYMERIZABLE COMPOSITIONS | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2020-11-26 | — | — | WO | disclosed |
| EP-3740543-A1 | INCREASED SATURATION OF ICE MELTING COMPOSITIONS AND METHODS OF USE | BASF SE (DE) | 2020-11-25 | — | — | EP | disclosed |
| US-20200339851-A1 | INCREASED SATURATION OF ICE MELTING COMPOSITIONS AND METHODS OF USE | BASF CORPORATION | 2020-10-29 | — | — | US | disclosed |
| US-20200315172-A1 | PEST CONTROL COMPOSITION INCLUDING NOVEL IMINOPYRIDINE DERIVATIVE | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2020-10-08 | — | — | US | disclosed |
| US-10736319-B2 | Pest control composition including novel iminopyridine derivative | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2020-08-11 | — | — | US | disclosed |
| WO-2020157598-A1 | ORTHODONTIC ARTICLES AND METHODS OF MAKING AND POSTPROCESSING SAME | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2020-08-06 | — | — | WO | disclosed |
| EP-3355933-B1 | ADENINE CONJUGATE COMPOUNDS AND THEIR USE AS VACCINE ADJUVANTS | SUMITOMO DAINIPPON PHARMA CO LTD (JP) | 2020-05-06 | — | — | EP | disclosed |
| US-10632192-B2 | Pyrimidine compounds and their use as vaccine adjuvants | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2020-04-28 | — | — | US | disclosed |
| US-20200121600-A1 | VACCINE ADJUVANT FORMULATION | Sumitomo Pharma Co., Ltd. (JP) | 2020-04-23 | — | — | US | disclosed |
| US-10597397-B2 | Adenine conjugate compounds and their use as vaccine adjuvants | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2020-03-24 | — | — | US | disclosed |
| EP-3603619-A1 | VACCINE ADJUVANT FORMULATION | Sumitomo Dainippon Pharma Co., Ltd. (JP) | 2020-02-05 | — | — | EP | disclosed |
| WO-2020003197-A2 | ORTHODONTIC ARTICLES PREPARED USING A POLYCARBONATE DIOL, POLYMERIZABLE COMPOSITIONS, AND METHODS OF MAKING THE ARTICLES | 3M INNOVATIVE PROPERTIES COMPANY (US) | 2020-01-02 | — | — | WO | disclosed |
| WO-2019141568-A1 | INCREASED SATURATION OF ICE MELTING COMPOSITIONS AND METHODS OF USE | BASF SE (DE) | 2019-07-25 | — | — | WO | disclosed |
| US-10349655-B2 | Pest control composition including novel iminopyridine derivative | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2019-07-16 | — | — | US | disclosed |
| US-20190200610-A1 | PEST CONTROL COMPOSITION INCLUDING NOVEL IMINOPYRIDINE DERIVATIVE | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2019-07-04 | — | — | US | disclosed |
| US-20180280499-A1 | PYRIMIDINE COMPOUND | Sumitomo Pharma Co., Ltd. (JP) | 2018-10-04 | — | — | US | disclosed |
| US-20180282334-A1 | ADENINE CONJUGATE COMPOUNDS AND THEIR USE AS VACCINE ADJUVANTS | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2018-10-04 | — | — | US | disclosed |
| EP-3355933-A1 | ADENINE CONJUGATE COMPOUNDS AND THEIR USE AS VACCINE ADJUVANTS | Sumitomo Dainippon Pharma Co., Ltd. (JP) | 2018-08-08 | — | — | EP | disclosed |
| US-20180042233-A1 | NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE HAVING 2-IMINO GROUP AND PEST CONTROL AGENT INCLUDING THE SAME | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2018-02-15 | — | — | US | disclosed |
| US-9758480-B2 | 1-(cycloalkyl-carbonyl)proline derivative | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2017-09-12 | — | — | US | disclosed |
| US-9718840-B2 | Condensed 5-oxazolidinone derivative | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2017-08-01 | — | — | US | disclosed |
| EP-2980067-B1 | PROCESSES FOR PREPARING OPTICALLY ACTIVE DIAMINE DERIVATIVES | DAIICHI SANKYO CO LTD (JP) | 2017-05-17 | — | — | EP | disclosed |
| EP-2634174-B1 | Nitrogen-containing heterocyclic derivate having 2-imino group and pest control agent including the same | MEIJI SEIKA PHARMA CO LTD (JP) | 2017-05-17 | — | — | EP | disclosed |
| EP-2907390-B1 | CONTROL AGENTS FOR HONEYBEE PARASITES AND CONTROL METHOD FOR HONEYBEE PARASITES USING SAME | MEIJI SEIKA PHARMA CO LTD (JP) | 2017-05-03 | — | — | EP | disclosed |
| US-20170022218-A1 | CONDENSED 5-OXAZOLIDINONE DERIVATIVE | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2017-01-26 | — | — | US | disclosed |
| EP-3095786-A1 | CONDENSED 5-OXAZOLIDINONE DERIVATIVE | Sumitomo Dainippon Pharma Co., Ltd. (JP) | 2016-11-23 | — | — | EP | disclosed |
| US-9447118-B2 | Preparation method of optically active diamine compound | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2016-09-20 | — | — | US | disclosed |
| US-20160165888-A1 | PEST CONTROL COMPOSITION INCLUDING NOVEL IMINOPYRIDINE DERIVATIVE | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2016-06-16 | — | — | US | disclosed |
| EP-1732931-B1 | METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO[2,3-b]FURAN-3-OL | JANSSEN SCIENCES IRELAND UC (IE) | 2016-05-18 | — | — | EP | disclosed |
| EP-1925611-B1 | OPTICALLY ACTIVE DIAMINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME | DAIICHI SANKYO CO LTD (JP) | 2016-04-13 | — | — | EP | disclosed |
| US-9301525-B2 | Pest control composition including novel iminopyridine derivative | MEUI SEIKA PHARMA CO., LTD. (JP) | 2016-04-05 | — | — | US | disclosed |
| EP-2980067-A1 | PROCESSES FOR PREPARING OPTICALLY ACTIVE DIAMINE DERIVATIVES | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2016-02-03 | — | — | EP | disclosed |
| US-20160016974-A1 | PREPARATION METHOD OF OPTICALLY ACTIVE DIAMINE COMPOUND | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2016-01-21 | — | — | US | disclosed |
| EP-2907390-A1 | CONTROL AGENTS FOR HONEYBEE PARASITES AND CONTROL METHOD FOR HONEYBEE PARASITES USING SAME | Meiji Seika Pharma Co., Ltd. (JP) | 2015-08-19 | — | — | EP | disclosed |
| US-20150210640-A1 | 1-(CYCLOALKYL-CARBONYL)PROLINE DERIVATIVE | SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) | 2015-07-30 | — | — | US | disclosed |
| US-9066517-B2 | Pest control agents for honeybee parasitic pests, and pest control method for honeybee parasitic pests using the pest control agents | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2015-06-30 | — | — | US | disclosed |
| EP-2876105-A1 | 1-(CYCLOALKYL-CARBONYL)PROLINE DERIVATIVE | Sumitomo Dainippon Pharma Co., Ltd. (JP) | 2015-05-27 | — | — | EP | disclosed |
| EP-2121679-B1 | METHOD FOR PRODUCING AZONIASPIRONORTROPINE ESTERS | K H S PHARMA HOLDING GMBH (DE) | 2015-04-15 | — | — | EP | disclosed |
| US-20150057288-A1 | PEST CONTROL AGENTS FOR HONEYBEE PARASITIC PESTS, AND PEST CONTROL METHOD FOR HONEYBEE PARASITIC PESTS USING THE PEST CONTROL AGENTS | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2015-02-26 | — | — | US | disclosed |
| US-20150005347-A1 | NITROGEN-CONTAINING HETEROCYCLIC DERIVATIVE HAVING 2-IMINO GROUP AND PEST CONTROL AGENT INCLUDING THE SAME | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2015-01-01 | — | — | US | disclosed |
| US-20140315839-A1 | PEST CONTROL COMPOSITION INCLUDING NOVEL IMINOPYRIDINE DERIVATIVE | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2014-10-23 | — | — | US | disclosed |
| US-8829208-B2 | Process for the preparation of darunavir and darunavir intermediates | MAPI PHARMA LTD. (IL) | 2014-09-09 | — | — | US | disclosed |
| US-8808961-B2 | Composition, resist film, pattern forming method, and inkjet recording method | FUJIFILM CORPORATION (JP) | 2014-08-19 | — | — | US | disclosed |
| EP-1211254-B1 | Process for the preparation of benzoxazine derivatives and intermediates therefor | DAIICHI SANKYO CO LTD (JP) | 2014-05-07 | — | — | EP | disclosed |
| EP-2284174-B1 | Intermediates for the preparation of benzoxazine derivatives and process for their preparation | DAIICHI SANKYO CO LTD (JP) | 2014-03-05 | — | — | EP | disclosed |
| EP-2025672-B1 | PROCESS FOR PRODUCING 1-CARBAMOYL-3,7-DIOXO-1,4-DIAZEPANE COMPOUNDS | DAIICHI SANKYO CO LTD (JP) | 2013-09-18 | — | — | EP | disclosed |
| WO-2013129688-A1 | PEST CONTROL COMPOSITION INCLUDING NOVEL IMINOPYRIDINE DERIVATIVE | MEIJI SEIKA PHARMA CO., LTD. (JP) | 2013-09-06 | — | — | WO | disclosed |
| EP-2634174-A2 | Nitrogen-containing hetercyclic derivate having 2-imino group and pest control agent including the same | Meiji Seika Pharma Co., Ltd. (JP) | 2013-09-04 | — | — | EP | disclosed |
| EP-2633756-A1 | Pest control composition including novel iminopyridine derivate | Meiji Seika Pharma Co., Ltd. (JP) | 2013-09-04 | — | — | EP | disclosed |
| EP-2360160-B1 | Intermediates and their use for producing benzoxazine derivative | DAIICHI SANKYO CO LTD (JP) | 2013-07-24 | — | — | EP | disclosed |
| EP-2218722-B9 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI SANKYO CO LTD (JP) | 2013-06-19 | — | — | EP | disclosed |
| EP-2218722-B1 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI SANKYO CO LTD (JP) | 2013-03-13 | — | — | EP | disclosed |
| EP-2528923-A1 | PROCESS FOR THE PREPARATION OF DARUNAVIR AND DARUNAVIR INTERMEDIATES | Mapi Pharma Limited (IL) | 2012-12-05 | — | — | EP | disclosed |
| US-20120296101-A1 | PROCESS FOR THE PREPARATION OF DARUNAVIR AND DARUNAVIR INTERMEDIATES | MAPI PHARMA LIMITED (IL) | 2012-11-22 | — | — | US | disclosed |
| EP-2477073-A1 | Resist composition for electron beam, EUV or X-ray | Fujifilm Corporation (JP) | 2012-07-18 | — | — | EP | disclosed |
| WO-2012063269-A2 | PROCESS FOR PREPARING ILOPERIDONE | CADILA HEALTHCARE LIMITED (IN) | 2012-05-18 | — | — | WO | disclosed |
| US-8163767-B2 | Heterocyclic Janus Kinase 3 inhibitors | ASTELLAS PHARMA INC. (JP) | 2012-04-24 | — | — | US | disclosed |
| EP-2130827-B1 | METHOD FOR PRODUCING QUINOLONE CARBOXYLIC ACID DERIVATIVE | DAIICHI SANKYO CO LTD (JP) | 2012-02-01 | — | — | EP | disclosed |
| US-8049006-B2 | 7-membered ring compound and method of production and pharmaceutical application thereof | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2011-11-01 | — | — | US | disclosed |
| EP-2360160-A1 | Intermediates and their use for producing benzoxazine derivative | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2011-08-24 | — | — | EP | disclosed |
| WO-2011092687-A1 | PROCESS FOR THE PREPARATION OF DARUNAVIR AND DARUNAVIR INTERMEDIATES | MAPI PHARMA HK LIMITED (CN) | 2011-08-04 | — | — | WO | disclosed |
| US-20110102528-A1 | COMPOSITION, RESIST FILM, PATTERN FORMING METHOD, AND INKJET RECORDING METHOD | FUJIFILM CORPORATION (JP) | 2011-05-05 | — | — | US | disclosed |
| US-20110065926-A1 | METHOD OF PREPARING IONIC LIQUIDS | BASF SE (DE) | 2011-03-17 | — | — | US | disclosed |
| US-7897806-B2 | Reacting primary amines with phosgene in ionic liquid as solvent | BASF AKTIENGESELLSCHAFT (DE) | 2011-03-01 | — | — | US | disclosed |
| EP-2284174-A1 | INTERMEDIATES FOR THE PREPARATION OF BENZOXAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION | Daiichi Sankyo Company, Limited (JP) | 2011-02-16 | — | — | EP | disclosed |
| US-7875722-B2 | having high antibacterial activity and high safety, at high yield and in a simple manner; one-pot process | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2011-01-25 | — | — | US | disclosed |
| US-7858802-B2 | Method of preparing ionic liquids | BASF SE (DE) | 2010-12-28 | — | — | US | disclosed |
| EP-2251341-A1 | Heterocyclic Janus kinase 3 inhibitors | Astellas Pharma Inc. (JP) | 2010-11-17 | — | — | EP | disclosed |
| EP-2218722-A2 | Process for producing benzoxazine derivative and production intermediate thereof | Daiichi Sankyo Company, Limited (JP) | 2010-08-18 | — | — | EP | disclosed |
| US-20100191010-A1 | PROCESS FOR THE SYNTHESIS OF CARBAMATES USING CO2 | HUNTSMAN INTERNATIONAL LLC (US) | 2010-07-29 | — | — | US | disclosed |
| EP-1435357-B1 | New process for the preparation of vinyl-pyrrolidinone cephalosporine derivatives | BASILEA PHARMACEUTICA AG (CH) | 2010-03-17 | — | — | EP | disclosed |
| US-20100063279-A1 | METHOD FOR PRODUCING QUINOLONE CARBOXYLIC ACID DERIVATIVE | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2010-03-11 | — | — | US | disclosed |
| US-20100048903-A1 | Method For Producing Azoniaspironortropine Esters And Nortropan-3-One Compounds | K.H.S. PHARMA HOLDING GMBH (DE) | 2010-02-25 | — | — | US | disclosed |
| EP-1448567-B1 | METHOD FOR THE PREPARATION OF HEXAHYDRO-FURO 2,3-B FURAN-3-OL | TIBOTEC PHARM LTD (IE) | 2009-12-30 | — | — | EP | disclosed |
| EP-2130827-A1 | METHOD FOR PRODUCING QUINOLONE CARBOXYLIC ACID DERIVATIVE | Daiichi Sankyo Company, Limited (JP) | 2009-12-09 | — | — | EP | disclosed |
| EP-2121679-A1 | METHOD FOR PRODUCING AZONIASPIRONORTROPINE ESTERS AND NORTROPAN-3-ONE COMPOUNDS | K.H.S. Pharma Holding Gmbh (DE) | 2009-11-25 | — | — | EP | disclosed |
| US-7612166-B2 | Fluorous capping reagents and methods for peptide purification | TRUSTEES OF TUFTS COLLEGE (US) | 2009-11-03 | — | — | US | disclosed |
| US-20090264399-A1 | HETEROCYCLIC JANUS KINASE 3 INHIBITORS | ASTELLAS PHARMA INC. (JP) | 2009-10-22 | — | — | US | disclosed |
| US-20090253683-A1 | 7-MEMBERED RING COMPOUND AND METHOD OF PRODUCTION AND PHARMACEUTICAL APPLICATION THEREOF | ASUBIO PHARMA CO., LTD (JP) | 2009-10-08 | — | — | US | disclosed |
| US-7595408-B2 | Methods for the preparation of (3R,3aS,6aR) hexahydro-furo[2,3-b]furan-3-ol | TIBOTEC PHARMACEUTICALS, LTD. (IE) | 2009-09-29 | — | — | US | disclosed |
| US-20090112017-A1 | METHOD FOR PRODUCING POLYISOCYANATES | BASF AKTIENGESSELLSCHAFT (DE) | 2009-04-30 | — | — | US | disclosed |
| US-20090105491-A1 | OPTICALLY ACTIVE DIAMINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME | DAIICHI SANKYO COMPANY, LIMITED (JP) | 2009-04-23 | — | — | US | disclosed |
| US-7521168-B2 | Compound that has a reduction potential higher than that of diphenyl iodonium salt and generates an acid upon irradiation of an actinic ray or radiation. | FUJIFILM CORPORATION (JP) | 2009-04-21 | — | — | US | disclosed |
| US-20090098447-A1 | RESIN COMPOSITION FOR FUEL CELL SEPARATOR, AND FUEL CELL SEPARATOR | NICHIAS CORPORATION (JP) | 2009-04-16 | — | — | US | disclosed |
| EP-2025672-A1 | SEVEN-MEMBERED RING COMPOUND, PRODUCTION METHOD THEREOF AND PHARMACEUTICAL USE THEREOF | Asubio Pharma Co., Ltd. (JP) | 2009-02-18 | — | — | EP | disclosed |
| EP-2011782-A1 | Process for the synthesis of carbamates using co2 | HUNTSMAN INTERNATIONAL LLC (US) | 2009-01-07 | — | — | EP | disclosed |
| US-20080275216-A1 | Fluorous Capping Reagents and Methods for Peptide Purification | TRUSTEES OF TUFTS COLLEGE (US) | 2008-11-06 | — | — | US | disclosed |
| WO-2008101728-A1 | METHOD FOR PRODUCING AZONIASPIRONORTROPINE ESTERS AND NORTROPAN-3-ONE COMPOUNDS | K.H.S. PHARMA HOLDING GMBH (DE) | 2008-08-28 | — | — | WO | disclosed |
| US-20080200535-A1 | sphingosine 1-phosphate-1/EDG-1 receptor agonists; autoimmune diseases; immunosuppressants by inducing lymphocyte sequestration in secondary lymphoid tissues; 4-aminocyclopentane-2-encarboxylic acid hydrochloric acid salt | ASAHI KASEI PHARMA CORPORATION (JP) | 2008-08-21 | — | — | US | disclosed |
| EP-1925611-A1 | OPTICALLY ACTIVE DIAMINE DERIVATIVE AND PROCESS FOR PRODUCING THE SAME | Daiichi Sankyo Company, Limited (JP) | 2008-05-28 | — | — | EP | disclosed |
| EP-1910358-A2 | HETEROCYCLIC JANUS KINASE 3 INHIBITORS | Astellas Pharma Inc. (JP) | 2008-04-16 | — | — | EP | disclosed |
| US-20070208184-A1 | METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO[2,3-b]FURAN-3-OL | Janssen Sciences Ireland Unlimited Company (IE) | 2007-09-06 | — | — | US | disclosed |
| US-20070142646-A1 | Method of preparing ionic liquids | BASF AKTIENGESELLSCHAFT (DE) | 2007-06-21 | — | — | US | disclosed |
| US-7189847-B2 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. (JP) | 2007-03-13 | — | — | US | disclosed |
| WO-2007007919-A2 | HETEROCYCLIC JANUS KINASE 3 INHIBITORS | ASTELLAS PHARMA INC. (JP) | 2007-01-18 | — | — | WO | disclosed |
| EP-1732931-A1 | METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO[2,3-b]FURAN-3-OL | Tibotec Pharmaceuticals Ltd. (IE) | 2006-12-20 | — | — | EP | disclosed |
| EP-1644395-B1 | PROCESSES FOR PREPARING 4'AZIDO NUCLEOSIDE DERIVATIVES | HOFFMANN LA ROCHE (CH) | 2006-11-22 | — | — | EP | disclosed |
| US-20060251961-A1 | Use of an ionic liquid | BASF AKTIENGESELLSCHAFT (DE) | 2006-11-09 | — | — | US | disclosed |
| US-7126015-B2 | Method for the preparation of hexahydro-furo-[2,3-b]furan-3-ol | TIBOTEC PHARMACEUTICALS LTD. (IE) | 2006-10-24 | — | — | US | disclosed |
| EP-1693704-A2 | Resist composition and pattern forming method using the same | Fuji Photo Film Co., Ltd. (JP) | 2006-08-23 | — | — | EP | disclosed |
| US-7087778-B2 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. (JP) | 2006-08-08 | — | — | US | disclosed |
| US-20060172226-A1 | Resist composition and pattern forming method using the same | FUJI PHOTO FILM CO., LTD. | 2006-08-03 | — | — | US | disclosed |
| US-20060167014-A1 | Piperazine compounds and medicinal use thereof | MITSUBISHI PHARMA CORPORATION | 2006-07-27 | — | — | US | disclosed |
| EP-1644395-A1 | PROCESSES FOR PREPARING 4'AZIDO NUCLEOSIDE DERIVATIVES | F. HOFFMANN-LA ROCHE AG (CH) | 2006-04-12 | — | — | EP | disclosed |
| US-20060014947-A1 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. | 2006-01-19 | — | — | US | disclosed |
| WO-2005118527-A2 | FLUOROUS CAPPING REAGENTS, AND METHODS FOR PEPTIDE PURIFICATION | TRUSTEES OF TUFTS COLLEGE (US) | 2005-12-15 | — | — | WO | disclosed |
| WO-2005095410-A1 | METHODS FOR THE PREPARATION OF (3R,3aS,6aR) HEXAHYDRO-FURO[2,3-b]FURAN-3-OL | TIBOTEC PHARMACEUTICALS LTD. (IE) | 2005-10-13 | — | — | WO | disclosed |
| EP-1029851-B1 | PIPERAZINE COMPOUNDS AND MEDICINAL USE THEREOF | MITSUBISHI PHARMA CORP (JP) | 2005-04-20 | — | — | EP | disclosed |
| EP-1289998-B1 | NEW PROCESS FOR THE PREPARATION OF VINYL-PYRROLIDINONE CEPHALOSPORINE DERIVATIVES | BASILEA PHARMACEUTICA AG (CH) | 2005-03-30 | — | — | EP | disclosed |
| US-6872823-B1 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. (JP) | 2005-03-29 | — | — | US | disclosed |
| US-20050038240-A1 | Processes for preparing 4'-azido-nucleoside derivatives | ROCHE PALO ALTO LLC | 2005-02-17 | — | — | US | disclosed |
| US-20050027119-A1 | Process for producing benzoxazine derivative and production intermediate thereof | DAIICHI PHARMACEUTICAL CO., LTD. | 2005-02-03 | — | — | US | disclosed |
| WO-2005000864-A1 | PROCESSES FOR PREPARING 4’AZIDO NUCLEOSIDE DERIVATIVES | F. HOFFMANN-LA ROCHE AG (CH) | 2005-01-06 | — | — | WO | disclosed |
| US-20040249175-A1 | Method for the preparation of hexahydro-furo-[2,3-b]furan-3-ol | Janssen Sciences Ireland Unlimited Company (IE) | 2004-12-09 | — | — | US | disclosed |
| EP-1448567-A1 | METHOD FOR THE PREPARATION OF HEXAHYDRO-FURO 2,3-B]FURAN-3-OL | Tibotec Pharmaceuticals Ltd. (IE) | 2004-08-25 | — | — | EP | disclosed |
| EP-1435357-A2 | New process for the preparation of vinyl-pyrrolidinone cephalosporine derivatives | Basilea Pharmaceutica AG (CH) | 2004-07-07 | — | — | EP | disclosed |
| EP-1027332-B1 | NOVEL LACTAM METALLOPROTEASE INHIBITORS | BRISTOL MYERS SQUIBB PHARMA CO (US) | 2004-05-26 | — | — | EP | disclosed |
| EP-1363890-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | Millennium Pharmaceuticals, Inc. (US) | 2003-11-26 | — | — | EP | disclosed |
| EP-1338921-A2 | Resist composition for electron beam, X-ray or EUV | Fuji Photo Film Co., Ltd. (JP) | 2003-08-27 | — | — | EP | disclosed |
| US-6610731-B2 | Antiinflammatory | BRISTOL-MYERS SQUIBB COMPANY | 2003-08-26 | — | — | US | disclosed |
| US-20030134827-A1 | Novel lactam metalloprotease inhibitors | DUAN JINGWU (US) | 2003-07-17 | — | — | US | disclosed |
| US-20030055064-A1 | Piperazine compounds and medicinal use thereof | MITSUBISHI PHARMA CORPORATION | 2003-03-20 | — | — | US | disclosed |
| WO-2003022853-A1 | METHOD FOR THE PREPARATION OF HEXAHYDRO-FURO[2,3-B]FURAN-3-OL | TIBOTEC PHARMACEUTICALS LTD. (IE) | 2003-03-20 | — | — | WO | disclosed |
| EP-1289998-A1 | NEW PROCESS FOR THE PREPARATION OF VINYL-PYRROLIDINONE CEPHALOSPORINE DERIVATIVES | Basilea Pharmaceutica AG (CH) | 2003-03-12 | — | — | EP | disclosed |
| US-20030018034-A1 | Piperazine compounds and medicinal use thereof | MITSUBISHI PHARMA CORPORATION | 2003-01-23 | — | — | US | disclosed |
| US-6504025-B2 | In fewer steps and is obtained in higher yield; chemical intermediates; useful in treating methicillin resistent Staphylococcus aureus and Pseudomonas aeruginosa | BASILEA PHARMACEUTICA AG (CH) | 2003-01-07 | — | — | US | disclosed |
| US-6455528-B1 | TUMOR NECROSIS FACTOR ANTAGONIST AND/OR INTERLEUKIN PROMOTER; ANTIALLERGENS, ANTIINFLAMMATORY AGENTS; AUTOIMMUNE DISEASE TREATMENT | MITSUBISHI PHARMA CORPORATION (JP) | 2002-09-24 | — | — | US | disclosed |
| WO-2002062766-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | MILLENNIUM PHARMACEUTICALS, INC. (US) | 2002-08-15 | — | — | WO | disclosed |
| WO-2002059118-A1 | PROCESS FOR N-(OXYALKYLATION) OF CARBOXAMIDES | SYNGENTA LIMITED (GB) | 2002-08-01 | — | — | WO | disclosed |
| US-6403632-B1 | CYCLIC AMIDE DERIVATIVE | BRISTOL MYERS SQUIBB PHARMA CO (US) | 2002-06-11 | — | — | US | disclosed |
| EP-1211254-A1 | PROCESS FOR THE PREPARATION OF BENZOXAZINE DERIVATIVES AND INTERMEDIATES THEREFOR | DAIICHI PHARMACEUTICAL CO., LTD. (JP) | 2002-06-05 | — | — | EP | disclosed |
| EP-1204645-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | Millennium Pharmaceuticals, Inc. (US) | 2002-05-15 | — | — | EP | disclosed |
| US-6372800-B1 | IMMUNOSUPPRESSIVE EFFECT AND IS USEFUL AS AN INHIBITOR FOR THE REJECTION REACTION OCCURRING IN ORGAN OR BONE MARROW TRANSPLANTATION, AND AS A PREVENTIVE OR REMEDY FOR ARTICULAR RHEUMATISM, ATOPIC ECZEMA (DERMATITIS), BEHCET'S DISEASE, | MITSUBISHI PHARMA CORPORATION (JP) | 2002-04-16 | — | — | US | disclosed |
| US-20020019381-A1 | Process for the preparation of vinyl-pyrrolidinone cephalosporin derivatives | BASILEA PHARMACEUTICA AG (CH) | 2002-02-14 | — | — | US | disclosed |
| EP-0778263-B1 | BENZENE COMPOUND AND MEDICINAL USE THEREOF | WELFIDE CORP (JP) | 2002-01-09 | — | — | EP | disclosed |
| WO-2001090111-A1 | NEW PROCESS FOR THE PREPARATION OF VINYL-PYRROLIDINONE CEPHALOSPORINE DERIVATIVES | BASILEA PHARMACEUTICA AG (CH) | 2001-11-29 | — | — | WO | disclosed |
| EP-0672718-B1 | Polyvinyl alcohol film, process for the production thereof and laminate | MITSUBISHI GAS CHEMICAL CO (JP) | 2001-06-06 | — | — | EP | disclosed |
| WO-2001010842-A2 | MELANOCORTIN-4 RECEPTOR BINDING COMPOUNDS AND METHODS OF USE THEREOF | MILLENNIUM PHARMACEUTICALS, INC. (US) | 2001-02-15 | — | — | WO | disclosed |
| US-6187821-B1 | SUCH AS 2-AMINO-2-(3-(4-HEPTYLPHENYL)PROPYL)BUTANE-1,4-DIOL; IMMUNOSUPPRESSANT; ADMINISTERING TO TREAT OR PREVENT AUTOIMMUNE DISEASES AND ALLERGIES | WELFIDE CORPORATION (JP) | 2001-02-13 | — | — | US | disclosed |
| EP-1029851-A1 | PIPERAZINE COMPOUNDS AND MEDICINAL USE THEREOF | YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) | 2000-08-23 | — | — | EP | disclosed |
| EP-1027332-A1 | NOVEL LACTAM METALLOPROTEASE INHIBITORS | Du Pont Pharmaceuticals Company (US) | 2000-08-16 | — | — | EP | disclosed |
| US-6057336-A | ANTIINFLAMMATORY AGENTS | E. I. DU PONT DE NEMOURS AND COMPANY (US) | 2000-05-02 | — | — | US | disclosed |
| US-6001851-A | HIV protease inhibitors | AGOURON PHARMACEUTICALS, INC. (US) | 1999-12-14 | — | — | US | disclosed |
| WO-1999018074-A1 | NOVEL LACTAM METALLOPROTEASE INHIBITORS | Britol-Myers Squibb Pharma Company (US) | 1999-04-15 | — | — | WO | disclosed |
| EP-0778263-A1 | BENZENE COMPOUND AND MEDICINAL USE THEREOF | YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) | 1997-06-11 | — | — | EP | disclosed |
| US-5582916-A | Polyvinyl alcohol film, process for the production thereof and laminate | MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) | 1996-12-10 | — | — | US | disclosed |
| EP-0672718-A1 | Polyvinyl alcohol film, process for the production thereof and laminate | MITSUBISHI GAS CHEMICAL COMPANY, INC. (JP) | 1995-09-20 | — | — | EP | disclosed |
| EP-0269042-B1 | PROCESS FOR PREPARING 2 PROPENYLIDENE-3 ETHYL GLUTARIC ACID DIESTERS | BASF Aktiengesellschaft (DE) | 1991-10-16 | — | — | EP | disclosed |
| US-4889911-A | ESTERIFICATION, ESTER INTERCHANGE; CATALYSIS WITH HETEROCYCLIC NITROGEN COMPOUND | BAYER AKTIENGESELLSCHAFT (DE) | 1989-12-26 | — | — | US | disclosed |
| US-4886869-A | OPTIONALLY SUBSTITUTED WITH-3-HYDROXY BENZOIC ACID; RIGIDITY, IMPACT STRENGTH AND ELONGATION | BAYER AKTIENGESELLSCHAFT (DE) | 1989-12-12 | — | — | US | disclosed |
| EP-0303931-A2 | Process for the fabrication of thermotropic, wholly aromatic polyesters and polyestercarbonates | BAYER AG (DE) | 1989-02-22 | — | — | EP | disclosed |
| EP-0303935-A2 | Thermotropic, aromatic polyestercarbonates, a process for their fabrication and their use | BAYER AG (DE) | 1989-02-22 | — | — | EP | disclosed |
| EP-0269042-A2 | Process for preparing 2 propenylidene-3 ethyl glutaric acid diesters | BASF Aktiengesellschaft (DE) | 1988-06-01 | — | — | EP | disclosed |
| EP-0269042-A2 | Process for preparing 2 propenylidene-3 ethyl glutaric acid diesters | BASF Aktiengesellschaft (DE) | 1988-06-01 | — | — | EP | disclosed |