SCHEMBL4832503

SCHEMBL4832503

CCC(CC)(C(=O)Oc1ccc(S(=O)(=O)NCC(=O)O)cc1)c1ccc(OC)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEP1B Q16820 1/20 0.49
MAPT P10636 1/20 0.46
TSHR P16473 1/20 0.46
ALDH1A1 P00352 7/20 0.45
PKM P14618 1/20 0.45
MMP1 P03956 4/20 0.44
GAA P10253 1/20 0.44
MMP12 P39900 1/20 0.44
MMP2 P08253 3/20 0.43
MMP13 P45452 3/20 0.43
ADAMTS4 O75173 1/20 0.43
MMP14 P50281 1/20 0.43
ADAMTS5 Q9UNA0 1/20 0.43
POLB P06746 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MMP9 P14780 2/20 0.42
MMP3 P08254 1/20 0.42
MMP7 P09237 1/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8657654 0.84 USP2 (0.49) MEP1BTSHRALDH1A1PKMPOLB
SCHEMBL4173740 0.83 MEP1B (0.67) MEP1BMAPTTSHRALDH1A1PKM
SCHEMBL8446269 0.75 MEP1B (0.58) MEP1BMAPTTSHRALDH1A1PKM
SCHEMBL4824911 0.74 HSD17B10 (0.67) MAPTALDH1A1GAAMMP2MMP13
SCHEMBL7383813 0.72 ALDH1A1 (0.71) MEP1BTSHRALDH1A1PKMMMP1
SCHEMBL6324179 0.72 MEP1B (0.67) MEP1BTSHRALDH1A1PKMMMP1
SCHEMBL27490403 0.70 NPC1 (0.46) ALDH1A1GAASMN1; SMN2MEN1LMNA
SCHEMBL5899469 0.70 ALDH1A1 (0.66) MEP1BMAPTTSHRALDH1A1PKM
SCHEMBL7345656 0.70 ALDH1A1 (0.62) MEP1BTSHRALDH1A1PKMMMP1
SCHEMBL8425825 0.69 MAPT (0.60) MEP1BMAPTALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US claimed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP claimed
US-7335686-B2 Method and composition for treating osteoporosis COUNCIL OF SCIENTIFIC AND INDUSTRIAL RESEARCH (IN) 2008-02-26 US disclosed
US-20050085537-A1 Method and composition for treating osteoporosis COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2005-04-21 US disclosed
US-6403644-B1 FOR PREVENTION AND/OR TREATMENT OF DISEASES INDUCED BY OVEREXPRESSION AND EXCESS ACTIVITY OF MATRIX METALLOPROTEINASE; FOR EXAMPLE, RHEUMATOID, ARTHROSTEITIS, UNUSUAL BONE RESORPTION, OSTEOPOROSIS, PERIODONTITIS ONO PHARMACEUTICAL CO., LTD. (JP) 2002-06-11 US disclosed
US-6177466-B1 Sulfonylamino acid derivatives ONO PHARMACEUTICAL CO., LTD. (JP) 2001-01-23 US disclosed
EP-0757037-A2 Sulfonylamino acid derivatives as metalloproteinase inhibitors ONO PHARMACEUTICAL CO., LTD. (JP) 1997-02-05 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050085537-A1 Method and composition for treating osteoporosis SOST, CALCR, MSR1 MEP1B 1893/4885MAPT 3941/4885TSHR 588/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.