SCHEMBL483716

SCHEMBL483716

CC(C)(C)OC(=O)N[C@@](C)(CCC(=O)c1cccc(OCc2ccccc2)c1)C(=O)O

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PTPN1 P18031 1/20 0.53
MAOB P27338 1/20 0.51
NR4A2 P43354 3/20 0.50
SMPD1 P17405 2/20 0.49
NR4A1 P22736 1/20 0.47
NR4A3 Q92570 1/20 0.47
GPR132 Q9UNW8 2/20 0.46
SRD5A2 P31213 1/20 0.46
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
NR1H4 Q96RI1 1/20 0.44
CYP19A1 P11511 1/20 0.44
FAAH O00519 1/20 0.44
CNR2 P34972 1/20 0.44
CTSK P43235 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL311818 0.89 EGFR (0.53) MAOBNR4A2NR4A1NR4A3SRD5A2
SCHEMBL483765 0.89 EGFR (0.53) MAOBNR4A2NR4A1NR4A3SRD5A2
SCHEMBL24310073 0.81 PTPN1 (0.55) PTPN1MAOBNR4A2SMPD1NR4A1
SCHEMBL2834205 0.81 GPR132 (0.55) PTPN1MAOBNR4A2GPR132CTSK
SCHEMBL483714 0.79 PTPN1 (0.50) PTPN1MAOBNR4A2SMPD1NR4A1
SCHEMBL310957 0.76 MAOB (0.51) PTPN1MAOBCTSK
SCHEMBL3350999 0.76 ITGB3 (0.55) PTPN1MAOBNR4A2NR4A1NR4A3
SCHEMBL840032 0.76 EGFR (0.50) MAOBNR4A2NR4A1NR4A3SRD5A2
SCHEMBL32665611 0.75 SMPD1 (0.60) PTPN1MAOBNR4A2SMPD1NR4A1
SCHEMBL2575501 0.75 CHRNA1 (0.38) MEN1KMT2ACTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8153623-B2 Compounds Convergence Pharmaceuticals Limited (GB) 2012-04-10 US disclosed
EP-1934176-B1 QUATERNARY ALPHA-AMINOCARBOXAMIDE DERIVATIVES AS MODULATORS OF VOLTAGE-GATED SODIUM CHANNELS GLAXO GROUP LTD (GB) 2012-02-01 EP disclosed