SCHEMBL4846089

SCHEMBL4846089

COc1ccc(C(=O)C=Cc2cc(-c3ccccc3OC)ccc2OCCN(C)C)cc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 1/20 0.55
TNFRSF1A P19438 3/20 0.54
ABCG2 Q9UNQ0 1/20 0.53
BCHE P06276 2/20 0.53
ACHE P22303 2/20 0.53
KEAP1 Q14145 1/20 0.51
NFE2L2 Q16236 1/20 0.51
RELA Q04206 2/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
MAPT P10636 2/20 0.48
KDM4E B2RXH2 2/20 0.48
LMNA P02545 1/20 0.48
ATM Q13315 1/20 0.48
L3MBTL1 Q9Y468 1/20 0.48
HTR7 P34969 1/20 0.48
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 1/20 0.47
RAB9A P51151 1/20 0.47
DPP4 P27487 2/20 0.47
PTPN1 P18031 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4853297 0.91 BCHE (0.52) MAOBTNFRSF1AABCG2BCHEACHE
SCHEMBL4851441 0.91 MAOB (0.54) MAOBTNFRSF1AABCG2BCHEACHE
SCHEMBL4849165 0.89 BCHE (0.58) MAOBTNFRSF1AABCG2BCHEACHE
SCHEMBL4850027 0.86 TNFRSF1A (0.47) TNFRSF1ABCHEACHERELASMN1; SMN2
SCHEMBL4848072 0.86 LMNA (0.48) TNFRSF1AABCG2RELASMN1; SMN2MAPT
SCHEMBL4854790 0.86 ABCG2 (0.50) TNFRSF1AABCG2SMN1; SMN2MAPTKDM4E
SCHEMBL5915495 0.84 HTR7 (0.53) MAOBTNFRSF1AABCG2BCHEKEAP1
SCHEMBL6386830 0.84 ABCG2 (0.52) MAOBTNFRSF1AABCG2BCHEACHE
SCHEMBL4845636 0.84 TNFRSF1A (0.49) TNFRSF1ABCHEACHESMN1; SMN2KDM4E
SCHEMBL4846085 0.84 TUBB4A (0.53) TNFRSF1AABCG2BCHEACHEMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US claimed
US-7423181-B2 in particular against bacterial and parasitic infections, fungi, and helminths; improved metabolic and physiochemical properties, bioavailability, solubility; 3-[4-(2-Dimethylamino-ethoxy)-2'-trifluoromethyl-biphenyl-3-yl]-1-(2-dimethylaminomethyl-phenyl)-propenone LICA PHARMACEUTICALS A/S (DK) 2008-09-09 US disclosed
US-20050227990-A1 Aminoalkoxy-functional chalcones LICA PHARMACEUTICALS A/S (DK) 2005-10-13 US disclosed