SCHEMBL4847559

SCHEMBL4847559

Nc1ncccc1NN1CCC(C(=O)O)CC1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NEK2 P51955 3/20 0.51
KDM4E B2RXH2 2/20 0.49
CYP2C19 P33261 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.44
ELANE P08246 1/20 0.44
SHMT2 P34897 1/20 0.44
GSK3B P49841 2/20 0.44
DYRK1A Q13627 2/20 0.41
ALDH1A1 P00352 1/20 0.40
NAPRT Q6XQN6 1/20 0.40
BACE1 P56817 1/20 0.38
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
ATR Q13535 1/20 0.38
MALT1 Q9UDY8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17506467 0.86 SHMT2 (0.46) NEK2KDM4ECYP2C19L3MBTL1ELANE
SCHEMBL2604305 0.76 BACE1 (0.40) ELANESHMT2GSK3BNAPRTBACE1
SCHEMBL4524152 0.73 NEK2 (0.67) NEK2KDM4ECYP2C19L3MBTL1ELANE
SCHEMBL7735744 0.71 L3MBTL1 (0.49) KDM4ECYP2C19L3MBTL1ALDH1A1
SCHEMBL788473 0.70 SHMT2 (0.44) KDM4EELANESHMT2GSK3BNAPRT
SCHEMBL308530 0.70 L3MBTL1 (0.47) NEK2KDM4ECYP2C19L3MBTL1GSK3B
SCHEMBL4137493 0.68 SHMT2 (0.66) KDM4ESHMT2GSK3BALDH1A1NAPRT
SCHEMBL2009115 0.67 ELANE (0.46) ELANEGSK3BALDH1A1
SCHEMBL2009118 0.67 ELANE (0.46) ELANEGSK3BALDH1A1
SCHEMBL17506389 0.67 SHMT2 (0.46) L3MBTL1ELANESHMT2GSK3BNAPRT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008070014-A2 BIARYL KETONE-SUBSTITUTED PIPERIDINES NEUROGEN CORPORATION (US) 2008-06-12 WO disclosed