SCHEMBL485961

SCHEMBL485961

Cc1cnccc1OC(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 2/20 0.43
SIRT3 Q9NTG7 1/20 0.43
SSTR4 P31391 1/20 0.40
POLB P06746 1/20 0.39
KDM4C Q9H3R0 2/20 0.37
CCNC P24863 2/20 0.36
CDK8 P49336 2/20 0.36
ALDH1A1 P00352 3/20 0.36
KDM4E B2RXH2 2/20 0.36
KMT2A Q03164 2/20 0.36
MEN1 O00255 1/20 0.36
KDM6B O15054 1/20 0.36
KDM4A O75164 1/20 0.36
MAPT P10636 1/20 0.36
THRB P10828 1/20 0.36
KDM4D Q6B0I6 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
GAA P10253 2/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9413729 0.85 TDP1 (0.47) TDP1SIRT3SSTR4POLBKDM4C
SCHEMBL21582000 0.83 SIRT3 (0.50) TDP1SIRT3SSTR4POLBKDM4C
SCHEMBL377258 0.82 ALDH1A1 (0.39) TDP1SIRT3KDM4CALDH1A1KDM4E
SCHEMBL27916164 0.80 ACHE (0.46) TDP1SIRT3SSTR4POLBALDH1A1
SCHEMBL7603934 0.78 CA12 (0.39) TDP1SIRT3KDM4CALDH1A1KDM4E
SCHEMBL4633528 0.77 ALDH1A1 (0.53) TDP1SIRT3KDM4CALDH1A1KDM4E
SCHEMBL9320822 0.77 GAA (0.41) TDP1KDM4CCCNCCDK8ALDH1A1
SCHEMBL9318384 0.76 SLC22A12 (0.51) KMT2A
SCHEMBL9413735 0.74 CYP2E1 (0.38) TDP1KDM4CCCNCCDK8ALDH1A1
SCHEMBL4633602 0.73 ALDH1A1 (0.48) TDP1SIRT3KDM4CALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2411363-B1 SUBSTITUTED PIPERIDINES AS PAR-1 ANTAGONISTS BAYER IP GMBH (DE) 2015-10-07 EP disclosed
EP-2411363-A1 SUBSTITUTED PIPERIDINES AS PAR-1 ANTAGONISTS Bayer Pharma AG (DE) 2012-02-01 EP disclosed
WO-2010108608-A1 SUBSTITUTED PIPERIDINES AS PAR-1 ANTAGONISTS BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2010-09-30 WO disclosed