SCHEMBL4865415

SCHEMBL4865415

COc1ccc(COC(=O)c2cn(N(CCNS(=O)(=O)c3nc4ccccc4s3)CC(=O)O)c(=O)nc2N)cc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.37
GLO1 Q04760 2/20 0.36
KEAP1 Q14145 1/20 0.35
NFE2L2 Q16236 1/20 0.35
MAPT P10636 5/20 0.35
GAA P10253 3/20 0.35
DHODH Q02127 2/20 0.34
KMT2A Q03164 4/20 0.34
MEN1 O00255 3/20 0.34
KDM4E B2RXH2 2/20 0.34
HPGD P15428 2/20 0.34
ALDH1A1 P00352 3/20 0.33
CA1 P00915 2/20 0.33
CA2 P00918 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4865411 0.84 ABL1 (0.41) PKMGLO1MAPTGAAKMT2A
SCHEMBL4839459 0.73 ABL1 (0.44) PKMGLO1MAPTGAAKMT2A
SCHEMBL4868081 0.69 CA1 (0.33) ALDH1A1CA1CA2
SCHEMBL4834952 0.68 PKM (0.33) PKMGLO1MAPTGAAKMT2A
SCHEMBL4838731 0.68 PKM (0.34) PKMGLO1MAPTGAAKMT2A
SCHEMBL3132617 0.68 ABL1 (0.41) PKMGLO1MAPTGAAKMT2A
SCHEMBL4404872 0.65 ABL1 (0.46) MAPTKMT2AMEN1KDM4EALDH1A1
SCHEMBL4838665 0.65 ABL1 (0.51) PKMGLO1MAPTKMT2AMEN1
SCHEMBL3140234 0.65 PAX8 (0.42) GLO1MAPTALDH1A1CA1CA2
SCHEMBL4868075 0.63 NPC1 (0.33) ALDH1A1CA1CA2SMN1; SMN2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7411065-B2 Peptide nucleic acid monomers: diphenylmethyl, benzyl, alkylthioalkyl, or phenylthioalkyl esters of N-(1-[4-(2-benzothiazolyl-, 2-benzoxazolyl-, 2-benzofuranyl- or 2-benzothiophenyl-sulfonyl)-3-piperazinon-1-ylcarbonylmethyl]pyrimidon-4-yl)carbamic acids PANAGENE, INC. (KR) 2008-08-12 US disclosed