SCHEMBL4874740

SCHEMBL4874740

CCOC(CN(C(=O)CC(=O)O)c1ccccc1)OCC

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.45
GLA P06280 1/20 0.45
TSHR P16473 1/20 0.45
TP53 P04637 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
OPRM1 P35372 4/20 0.39
NPC1 O15118 1/20 0.38
JAK2 O60674 1/20 0.38
RAB9A P51151 1/20 0.38
PAX8 Q06710 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
HPGD P15428 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4865282 0.88 SMN1; SMN2 (0.43) ALDH1A1GLATSHRTP53SMN1; SMN2
SCHEMBL4874004 0.88 ALDH1A1 (0.42) ALDH1A1GLATSHRTP53SMN1; SMN2
SCHEMBL308738 0.79 ALDH1A1 (0.66) ALDH1A1GLATSHRTP53SMN1; SMN2
SCHEMBL8303367 0.76 HTT (0.52) ALDH1A1SMN1; SMN2MEN1KMT2AOPRM1
SCHEMBL3583408 0.76 TP53 (0.43) ALDH1A1GLATSHRTP53SMN1; SMN2
SCHEMBL11063095 0.73 ALDH1A1 (0.44) ALDH1A1SMN1; SMN2KMT2AOPRM1NPC1
SCHEMBL7238334 0.73 KDM4E (0.41) ALDH1A1GLATSHRTP53MEN1
SCHEMBL11065640 0.72 ALDH1A1 (0.43) ALDH1A1TP53NPC1RAB9ACYP3A4
SCHEMBL11062234 0.72 ALDH1A1 (0.43) ALDH1A1OPRM1NPC1RAB9AHPGD
SCHEMBL11065506 0.72 L3MBTL1 (0.50) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7442693-B2 Diazepine compounds as ligands of the melanocortin 1 and/or 4 receptors SMITHKLINE BEECHAM CORPORATION (US) 2008-10-28 US disclosed
US-20070270411-A1 Novel Diazepine Compounds as Ligands of the Melanocortin 1 and/or 4 Receptors SMITHKLINE BEECHAM CORPORATION 2007-11-22 US disclosed
WO-2005118573-A1 NOVEL DIAZEPINE COMPOUNDS AS LIGANDS OF THE MELANOCORTIN 1 AND/OR 4 RECEPTORS SMITHKLINE BEECHAM CORPORATION (US) 2005-12-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070270411-A1 Novel Diazepine Compounds as Ligands of the Melanocortin 1 and/or 4 Receptors MC4R, MC3R, MC5R ALDH1A1 2986/4885GLA 4736/4885TSHR 203/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.