SCHEMBL4882778

SCHEMBL4882778

Fc1ccc(-n2nc[c]c2C(F)(F)F)cc1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.39
CYP1A2 P05177 1/20 0.39
NR3C1 P04150 8/20 0.39
PGR P06401 2/20 0.39
KDM4E B2RXH2 2/20 0.37
SRC P12931 1/20 0.37
BRAF P15056 1/20 0.37
KDR P35968 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
LMNA P02545 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PTGS2 P35354 4/20 0.34
PTGS1 P23219 4/20 0.34
XDH P47989 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16927650 0.87 XDH (0.44) KDM4ESRCBRAFKDRNPSR1
SCHEMBL1304888 0.84 NPBWR1 (0.39) CYP1A2NR3C1NPSR1LMNAMEN1
SCHEMBL885439 0.84 PTGS1 (0.43) CYP1A2KDM4ENPSR1LMNAPTGS2
SCHEMBL219809 0.84 SMN1; SMN2 (0.41) CYP1A2KDM4EBRAFNPSR1LMNA
SCHEMBL16927664 0.80 PTGS2 (0.47) CYP1A2NPSR1LMNAKMT2APTGS2
SCHEMBL16927613 0.80 NPBWR1 (0.39) KDM4E
SCHEMBL28417582 0.80 POLB (0.41) CYP17A1CYP1A2LMNAMEN1KMT2A
SCHEMBL15016131 0.78 PTGS1 (0.46) NPSR1MEN1KMT2APTGS2PTGS1
SCHEMBL16927635 0.78 PTGS2 (0.47) CYP1A2PTGS2PTGS1
SCHEMBL16927593 0.77 CYP17A1 (0.38) CYP17A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111362934-A Isothiazole oxadiazole derivatives, and preparation method and application thereof 南开大学 2020-07-03 CN claimed
CN-111362934-A Isothiazole oxadiazole derivatives, and preparation method and application thereof 南开大学 2020-07-03 CN disclosed
EP-2342196-B1 PYRAZOLE COMPOUNDS FOR CONTROLLING INVERTEBRATE PESTS BASF SE (DE) 2015-07-29 EP disclosed
US-20080064690-A1 PYRAZOLE-AMIDES AND -SULFONAMIDES ICAGEN, INC. (US) 2008-03-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080064690-A1 PYRAZOLE-AMIDES AND -SULFONAMIDES SCN3A, TRPV3, HCN3 CYP17A1 4637/4885CYP1A2 1874/4885NR3C1 3261/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.