SCHEMBL489171

SCHEMBL489171

CCC(OC(C)=O)(c1ccccc1)C(CC(C)NC)c1ccccc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR1 P21554 3/20 0.35
CNR2 P34972 3/20 0.35
KCNH2 Q12809 4/20 0.35
CHRM3 P20309 2/20 0.35
ADRA1A P35348 2/20 0.35
OPRK1 P41145 2/20 0.35
OPRM1 P35372 2/20 0.35
OPRD1 P41143 2/20 0.35
MRGPRX2 Q96LB1 1/20 0.35
HRH2 P25021 1/20 0.35
HTR2A P28223 1/20 0.35
CACNA1F O60840 1/20 0.35
CHRM2 P08172 1/20 0.35
CHRM1 P11229 1/20 0.35
ADRA2B P18089 1/20 0.35
HRH1 P35367 1/20 0.35
CACNA1D Q01668 1/20 0.35
SLC6A3 Q01959 1/20 0.35
CACNA1S Q13698 1/20 0.35
CACNA1C Q13936 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4972971 0.78 KCNH2 (0.44) KCNH2CHRM3ADRA1AOPRK1OPRM1
SCHEMBL4638235 0.72 KIF11 (0.39) KCNH2CHRM3ADRA1AOPRK1OPRM1
SCHEMBL5861679 0.71 KIF11 (0.38) KCNH2CHRM3ADRA1AOPRK1OPRM1
SCHEMBL7281996 0.67 HRH1 (0.62) CNR1KCNH2CHRM3ADRA1AOPRK1
Hydrochloric Acid SCHEMBL7274257 0.65 HRH1 (0.60) CNR1KCNH2CHRM3ADRA1AOPRK1
SCHEMBL10234508 0.64 CYP2C19 (0.46) KCNH2CHRM3OPRM1CHRM2CHRM1
SCHEMBL18994323 0.64 OPRM1 (0.64) KCNH2CHRM3OPRK1OPRM1OPRD1
SCHEMBL6014665 0.64 OPRM1 (0.64) KCNH2CHRM3OPRK1OPRM1OPRD1
SCHEMBL11530 0.64 CYP2D6 (0.40) KCNH2CHRM3ADRA1AOPRK1OPRM1
SCHEMBL7374412 0.63 KCNH2 (0.47) KCNH2CHRM3ADRA1AOPRK1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 545 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240288374-A1 PLASMONIC NANOPARTICLE PLATFORM FOR ANALYTE DETECTION Zymeron Corporation 2024-08-29 US claimed
WO-2024172892-A1 PLASMONIC NANOPARTICLE PLATFORM FOR ANALYTE DETECTION Zymeron Corporation (US) 2024-08-22 WO claimed
US-20150313846-A1 PROLONGED-RELEASE MULTIMICROPARTICULATE ORAL PHARMACEUTICAL FORM FLAMEL IRELAND LIMITED (IE) 2015-11-05 US claimed
US-9023400-B2 Prolonged-release multimicroparticulate oral pharmaceutical form FLAMEL TECHNOLOGIES (FR) 2015-05-05 US claimed
US-9016221-B2 Surface topographies for non-toxic bioadhesion control UNIVERSITY OF FLORIDA RESEARCH FOUNDATION, INC. (US) 2015-04-28 US claimed
US-8895063-B2 Oral dosage form comprising an antimisuse system FLAMEL TECHNOLOGIES (FR) 2014-11-25 US claimed
WO-2014153099-A2 METHOD FOR USING EXHALED BREATH TO DETERMINE THE PRESENCE OF DRUG Pulmonary Analytics (US) 2014-09-25 WO claimed
US-20140288454-A1 Method For Using Exhaled Breath to Determine the Presence of Drug Pulmonary Analytics (US) 2014-09-25 US claimed
US-8652529-B2 Anti-misuse microparticulate oral pharmaceutical form FLAMEL TECHNOLOGIES (FR) 2014-02-18 US claimed
US-8445023-B2 Anti-misuse microparticulate oral pharmaceutical form FLAMEL TECHNOLOGIES (FR) 2013-05-21 US claimed
WO-2006089843-A2 ANTI-MISUSE MICROPARTICULATE ORAL DRUG FORM FLAMEL TECHNOLOGIES (FR) 2006-08-31 WO claimed
EP-1569925-A1 2-SUBSTITUTED QUINAZOLIN-4-YLAMINE ANALOGUES AS CAPSAICIN RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2005-09-07 EP claimed
WO-2004055003-A1 2-SUBSTITUTED QUINAZOLIN-4-YLAMINE ANALOGUES AS CAPSAICIN RECEPTOR MODULATORS NEUROGEN CORPORATION (US) 2004-07-01 WO claimed
WO-2004028548-A2 INHIBITORS OF THE NITRIX OXIDE SYNTHASE III (NOS III) AS NEUROPROTECTIVE AGENTS CARBOMER, INC. (US) 2004-04-08 WO claimed
US-20040063612-A1 Neuroprotective agents CARBOMER, INC. 2004-04-01 US claimed
EP-0608893-B1 Compositions for inhibiting the development of tolerance to and/or dependence on an additive substance UNIV VIRGINIA COMMONWEALTH (US) 2001-12-12 EP claimed
US-5654281-A Inhibiting the development of tolerance to and/or dependence on an addictive substance VIRGINIA COMMONWEALTH UNIVERSITY (US) 1997-08-05 US claimed
EP-0608893-A1 Inhibiting the development of tolerance to and/or dependence on an additive substance VIRGINIA COMMONWEALTH UNIVERSITY (US) 1994-08-03 EP claimed
EP-0174342-B1 BRAIN-SPECIFIC ANALOGUES OF CENTRALLY ACTING AMINES UNIVERSITY OF FLORIDA (US) 1989-12-20 EP claimed
US-4126684-A 4-AMINO-3-P-HALOPHENYLBUTYRIC ACIDS AND THEIR DERIVATIVES USED IN THE CONTROL OF NARCOTIC ABUSE CIBA-GEIGY CORPORATION (US) 1978-11-21 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040063612-A1 Neuroprotective agents GAP43, NLN, NOS3 CNR1 1532/4885CNR2 1846/4885KCNH2 2862/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.