SCHEMBL4893199

SCHEMBL4893199

O=C(O)[C@@H]1CCCN1C(=O)c1ccncc1

nearest known ligand 0.62

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CA2 P00918 1/20 0.62
ALDH1A1 P00352 3/20 0.60
L3MBTL1 Q9Y468 2/20 0.56
TDP1 Q9NUW8 1/20 0.56
NPSR1 Q6W5P4 1/20 0.53
RECQL P46063 1/20 0.52
KDM4E B2RXH2 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3143281 1.00 CA2 (0.62) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL7960313 0.95 TDP1 (0.61) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL5537767 0.89 CA2 (0.75) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL6787910 0.89 CA2 (0.75) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL28789388 0.85 CA2 (0.67) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL13229 0.85 CA2 (0.67) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL13230 0.85 CA2 (0.67) CA2ALDH1A1L3MBTL1TDP1NPSR1
SCHEMBL4893223 0.82 ALDH1A1 (0.66) CA2ALDH1A1L3MBTL1
SCHEMBL2226530 0.82 ALDH1A1 (0.66) CA2ALDH1A1L3MBTL1
SCHEMBL13804351 0.82 GAA (0.53) L3MBTL1TDP1RECQLKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080200512-A1 Hepatitis C virus polymerase inhibitors BLANEY JEFFREY MARK 2008-08-21 US disclosed
US-6867211-B2 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy MERCKLE GMBH (DE) 2005-03-15 US disclosed
EP-1252163-B1 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2003-09-24 EP disclosed
US-20030153558-A1 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy MERCKLE GMBH (DE) 2003-08-14 US disclosed
EP-1252163-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2002-10-30 EP disclosed
WO-2001057042-A2 4-PYRIDYL-AND 2,4-PYRIMIDINYL-SUBSTITUTED PYRROLE DERIVATIVES AND THEIR USE IN PHARMACY MERCKLE GMBH (DE) 2001-08-09 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080200512-A1 Hepatitis C virus polymerase inhibitors SSU72, POLR2H, POLR2E CA2 1113/4885ALDH1A1 276/4885L3MBTL1 3221/4885
US-20030153558-A1 4-Pyridyl-and 2,4-pyrimidinyl-substituted pyrrole derivatives and their use in pharmacy IL4, IL2, IL5 CA2 3163/4885ALDH1A1 524/4885L3MBTL1 4875/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.