SCHEMBL4901779

SCHEMBL4901779

O=S(=O)(c1cc(Cl)c(O)c(Cl)c1)N1CCOc2ccccc21

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.57
POLB P06746 2/20 0.49
NR1H3 Q13133 2/20 0.48
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 1/20 0.46
NAMPT P43490 1/20 0.44
CPT2 P23786 1/20 0.43
CPT1A P50416 1/20 0.43
HTR6 P50406 3/20 0.42
CYP2C9 P11712 2/20 0.42
RORC P51449 1/20 0.42
NR1H2 P55055 1/20 0.42
PKM P14618 2/20 0.42
JAK2 O60674 1/20 0.42
NOTUM Q6P988 1/20 0.42
MAPT P10636 1/20 0.41
PKLR P30613 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1191891 0.83 SLC22A6 (0.47) NPC1NR1H3MEN1KMT2AALDH1A1
SCHEMBL3000456 0.81 NPC1 (0.59) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL5474787 0.80 NPC1 (0.58) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL2995685 0.80 NPC1 (0.58) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL3001581 0.77 VCAM1 (0.55) NPC1POLBMEN1KMT2AALDH1A1
SCHEMBL16217090 0.76 NPC1 (0.74) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL25442268 0.75 NPC1 (0.69) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL31750670 0.75 NPC1 (0.62) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL25754848 0.75 NPC1 (0.62) NPC1POLBNR1H3MEN1KMT2A
SCHEMBL25166791 0.74 NPC1 (0.67) NPC1POLBNR1H3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080064871-A1 Production Method of Nitrogen-Containing Fused Ring Compounds JAPAN TOBACCO INC. (JP) 2008-03-13 US claimed
EP-1820515-A1 NITROGEN-CONTAINING FUSED RING COMPOUND AND USE THEREOF Japan Tobacco, Inc. (JP) 2007-08-22 EP claimed
US-20070010670-A1 Nitrogen-containing fused ring compounds and use thereof JAPAN TOBACCO INC. (JP) 2007-01-11 US claimed
US-20080305169-A1 Pharmaceutical Compositions Comprising Nitrogen-Containing Fused Ring Coumpounds JAPAN TOBACCO INC. (JP) 2008-12-11 US disclosed
US-20080305169-A1 Pharmaceutical Compositions Comprising Nitrogen-Containing Fused Ring Coumpounds JAPAN TOBACCO INC. (JP) 2008-12-11 US disclosed
US-20080305169-A1 Pharmaceutical Compositions Comprising Nitrogen-Containing Fused Ring Coumpounds JAPAN TOBACCO INC. (JP) 2008-12-11 US disclosed
US-20080064871-A1 Production Method of Nitrogen-Containing Fused Ring Compounds JAPAN TOBACCO INC. (JP) 2008-03-13 US disclosed
US-20080064871-A1 Production Method of Nitrogen-Containing Fused Ring Compounds JAPAN TOBACCO INC. (JP) 2008-03-13 US disclosed
US-20080064871-A1 Production Method of Nitrogen-Containing Fused Ring Compounds JAPAN TOBACCO INC. (JP) 2008-03-13 US disclosed
EP-1820515-A1 NITROGEN-CONTAINING FUSED RING COMPOUND AND USE THEREOF Japan Tobacco, Inc. (JP) 2007-08-22 EP disclosed
US-20070010670-A1 Nitrogen-containing fused ring compounds and use thereof JAPAN TOBACCO INC. (JP) 2007-01-11 US disclosed
US-20070010670-A1 Nitrogen-containing fused ring compounds and use thereof JAPAN TOBACCO INC. (JP) 2007-01-11 US disclosed
US-20070010670-A1 Nitrogen-containing fused ring compounds and use thereof JAPAN TOBACCO INC. (JP) 2007-01-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080305169-A1 Pharmaceutical Compositions Comprising Nitrogen-Containing Fused Ring Coumpounds NOD1, NLRP3, SLC10A1 NPC1 145/4885POLB 4604/4885NR1H3 249/4885
US-20070010670-A1 Nitrogen-containing fused ring compounds and use thereof NUDT1, NOD1, SLC28A1 NPC1 489/4885POLB 4164/4885NR1H3 760/4885
US-20080064871-A1 Production Method of Nitrogen-Containing Fused Ring Compounds NOD1, XDH, URB2 NPC1 924/4885POLB 4495/4885NR1H3 681/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.