SCHEMBL4902965

SCHEMBL4902965

CCn1c(COCc2ccccc2)nc(C2CC2)c1I

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.38
ADORA2A P29274 1/20 0.37
ADORA1 P30542 1/20 0.37
AVPR1A P37288 1/20 0.35
VCP P55072 1/20 0.35
ALDH1A1 P00352 2/20 0.35
HPGD P15428 1/20 0.35
HTT P42858 1/20 0.35
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
ACSS2 Q9NR19 2/20 0.34
CCR2 P41597 1/20 0.33
NPC1 O15118 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2D6 P10635 1/20 0.33
MAPT P10636 1/20 0.33
CYP2C19 P33261 1/20 0.33
RAB9A P51151 1/20 0.33
SOAT1 P35610 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4901487 0.89 MEN1 (0.36) ADORA2AADORA1ALDH1A1MEN1KMT2A
SCHEMBL4900968 0.78 ALDH1A1 (0.48) TSHRALDH1A1HTTMEN1KMT2A
SCHEMBL4902092 0.74 TSHR (0.35) TSHRADORA2AADORA1AVPR1AALDH1A1
SCHEMBL4902069 0.69 TSHR (0.46) TSHRALDH1A1HTTKMT2ANPC1
SCHEMBL4899447 0.69 TSHR (0.42) TSHRADORA2AADORA1CCR2SOAT1
SCHEMBL17895924 0.66 AGTR1 (0.43) TSHRVCPALDH1A1HPGDMEN1
SCHEMBL22322658 0.64 KMT2A (0.44) TSHRVCPALDH1A1HPGDMEN1
SCHEMBL31085266 0.63 TSHR (0.36) TSHRADORA1VCPALDH1A1HTT
SCHEMBL23261777 0.63 VCP (0.36) TSHRVCPALDH1A1KMT2ACYP1A2
Propane SCHEMBL11584021 0.63 TSHR (0.83) TSHRALDH1A1MAPTPOLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080132549-A1 Sulphur-Linked Imidazone Compounds for the Treatment of Hiv/Aids PFIZER INC. (US) 2008-06-05 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080132549-A1 Sulphur-Linked Imidazone Compounds for the Treatment of Hiv/Aids SPR, TPMT, IMPDH1 TSHR 3874/4885ADORA2A 4532/4885ADORA1 3505/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.