SCHEMBL4906498

SCHEMBL4906498

O=P(O)(O)OCc1ccc(P(=O)(O)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.48
AKR1C3 P42330 1/20 0.44
CA2 P00918 1/20 0.43
CA4 P22748 1/20 0.43
CA5A P35218 1/20 0.43
CETP P11597 3/20 0.38
PDPK1 O15530 2/20 0.37
MTOR P42345 1/20 0.37
ALPG P10696 1/20 0.37
PTK2B Q14289 1/20 0.37
S1PR1 P21453 2/20 0.36
S1PR3 Q99500 2/20 0.36
PTPN2 P17706 3/20 0.35
PTPN1 P18031 3/20 0.35
PTPN6 P29350 3/20 0.35
PTPRC P08575 2/20 0.35
PTPRB P23467 2/20 0.35
PTPN11 Q06124 2/20 0.35
CDC25A P30304 1/20 0.35
SRC P12931 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17345002 0.89 TSHR (0.58) TSHRAKR1C3CETPPDPK1MTOR
SCHEMBL8384625 0.83 TSHR (0.52) TSHRAKR1C3CA2CETPPTPN1
SCHEMBL28365963 0.81 TSHR (0.50) TSHRAKR1C3CA2CA4CA5A
SCHEMBL31091007 0.79 TSHR (0.48) TSHRAKR1C3S1PR1S1PR3PTPN2
SCHEMBL207268 0.79 RAB9A (0.53) TSHRAKR1C3CA2S1PR1S1PR3
SCHEMBL27541457 0.79 TSHR (0.48) TSHRAKR1C3MEN1KMT2A
SCHEMBL19917829 0.79 TSHR (0.48) TSHRAKR1C3CETPPDPK1MTOR
SCHEMBL12786033 0.79 TSHR (0.48) TSHRAKR1C3CA2S1PR1S1PR3
SCHEMBL9093550 0.79 FDPS (0.50) TSHRAKR1C3CETPS1PR1S1PR3
SCHEMBL206610 0.78 TSHR (0.76) TSHRCETPPDPK1MTORALPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080200679-A1 Alpha-HYDROXY, alpha-SUBSTITUTED METHYLENEBISPHOSPHONATES AND PHOSPHONOACETATES UNIVERSITY OF SOUTHERN CALIFORNIA (US) 2008-08-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080200679-A1 Alpha-HYDROXY, alpha-SUBSTITUTED METHYLENEBISPHOSPHONATES AND PHOSPHONOACETATES GRHPR, PHPT1, PHYKPL TSHR 3136/4885AKR1C3 1160/4885CA2 2530/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.