SCHEMBL4910951

SCHEMBL4910951

N#Cc1ccccc1OCC(=O)Nc1ccccc1C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.59
GAA P10253 2/20 0.59
TRPM4 Q8TD43 2/20 0.58
MAPK1 P28482 1/20 0.57
NOTUM Q6P988 1/20 0.57
HCAR2 Q8TDS4 3/20 0.56
KMT2A Q03164 3/20 0.55
MEN1 O00255 2/20 0.55
CASP3 P42574 1/20 0.55
SENP8 Q96LD8 1/20 0.55
SENP7 Q9BQF6 1/20 0.55
SENP6 Q9GZR1 1/20 0.55
ALDH1A1 P00352 3/20 0.55
NPC1 O15118 5/20 0.55
RAB9A P51151 5/20 0.55
KDM4E B2RXH2 3/20 0.54
POLB P06746 2/20 0.54
TP53 P04637 1/20 0.53
NPSR1 Q6W5P4 1/20 0.53
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13744249 0.82 NOTUM (0.74) SMN1; SMN2GAAMAPK1NOTUMKMT2A
SCHEMBL8689307 0.81 HCAR2 (0.72) SMN1; SMN2GAATRPM4HCAR2KMT2A
SCHEMBL5150684 0.80 MEN1 (0.72) SMN1; SMN2TRPM4MAPK1NOTUMHCAR2
SCHEMBL4912967 0.80 TRPM4 (0.77) SMN1; SMN2GAATRPM4HCAR2KMT2A
SCHEMBL8689335 0.80 HSD17B10 (0.77) SMN1; SMN2GAAHCAR2KMT2AMEN1
SCHEMBL8689129 0.80 HCAR2 (0.60) SMN1; SMN2TRPM4NOTUMHCAR2KMT2A
SCHEMBL4913355 0.80 L3MBTL1 (0.64) SMN1; SMN2TRPM4HCAR2KMT2AMEN1
SCHEMBL26334075 0.79 SMN1; SMN2 (0.69) SMN1; SMN2GAAMAPK1NOTUMKMT2A
SCHEMBL5696401 0.79 KDM4E (0.64) SMN1; SMN2TRPM4MAPK1HCAR2KMT2A
SCHEMBL6032429 0.78 HCAR2 (0.81) SMN1; SMN2HCAR2KMT2AMEN1CASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2008-10-30 US claimed
US-7408078-B2 Anthranilic acid derivatives useful in treating infection with hepatitis C virus WYETH (US) 2008-08-05 US claimed
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus VIROPHARMA INCORPORATED 2005-01-06 US claimed
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2008-10-30 US disclosed
US-7408078-B2 Anthranilic acid derivatives useful in treating infection with hepatitis C virus WYETH (US) 2008-08-05 US disclosed
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus VIROPHARMA INCORPORATED 2005-01-06 US disclosed
WO-2004091724-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS WYETH (US) 2004-10-28 WO disclosed
US-5741926-A ANTIDIABETIC AGENT SHAMAN PHARMACEUTICALS, INC. (US) 1998-04-21 US disclosed
WO-1997030019-A1 ANILINE DERIVATIVES HAVING ANTIHYPERGLYCEMIC ACTIVITY SHAMAN PHARMACEUTICALS, INC. (US) 1997-08-21 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050004192-A1 Anthranilic acid derivatives useful in treating infection with hepatitis C virus HCCS, ALAD, HAVCR2 SMN1; SMN2 4765/4885GAA 212/4885TRPM4 4134/4885
US-20080269333-A1 ANTHRANILIC ACID DERIVATIVES USEFUL IN TREATING INFECTION WITH HEPATITIS C VIRUS HCCS, ALAD, HAVCR2 SMN1; SMN2 4765/4885GAA 212/4885TRPM4 4134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.