SCHEMBL4920244

SCHEMBL4920244

O=S(=O)(Nc1cncc(-c2ccncc2)c1)c1ccc(Cl)cc1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.66
ALPL P05186 6/20 0.63
CYP3A4 P08684 2/20 0.58
CYP2D6 P10635 2/20 0.58
PSEN1 P49768 1/20 0.58
PSEN2 P49810 1/20 0.58
APH1B Q8WW43 1/20 0.58
NCSTN Q92542 1/20 0.58
APH1A Q96BI3 1/20 0.58
PSENEN Q9NZ42 1/20 0.58
PIK3CA P42336 2/20 0.57
PIK3CG P48736 2/20 0.57
PIK3CD O00329 1/20 0.57
HTT P42858 1/20 0.56
PIK3CB P42338 4/20 0.53
CES1 P23141 1/20 0.53
CYP19A1 P11511 1/20 0.51
F2 P00734 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15211823 0.78 ALPL (1.00) ALPL
SCHEMBL4931253 0.76 XDH (0.56) ALPLCYP3A4CYP2D6PSEN1PSEN2
SCHEMBL9568492 0.75 KMT2A (0.72) ALDH1A1ALPLCYP3A4CYP2D6HTT
SCHEMBL3665383 0.74 PIK3CG (1.00) PIK3CAPIK3CGPIK3CDPIK3CB
SCHEMBL16529326 0.74 CYP3A4 (0.56) ALDH1A1CYP3A4CYP2D6PSEN1PSEN2
SCHEMBL30828581 0.73 ALDH1A1 (0.73) ALDH1A1CYP3A4CYP2D6PSEN1PSEN2
Hydrochloric Acid SCHEMBL939057 0.73 PIK3CG (0.98) PIK3CAPIK3CGPIK3CDPIK3CB
SCHEMBL2118369 0.73 ALDH1A1 (0.56) ALDH1A1CYP3A4CYP2D6PSEN1PSEN2
SCHEMBL4195479 0.73 APP (0.61) ALDH1A1CYP3A4CYP2D6PSEN1PSEN2
SCHEMBL14689318 0.72 MEN1 (0.60) ALDH1A1PIK3CACES1CYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080194584-A1 Nitrogen Heteroaromatic Compounds Which Bind To The Active Site Of Protein Kinase Enzymes GALAPAGOS NV (BE) 2008-08-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080194584-A1 Nitrogen Heteroaromatic Compounds Which Bind To The Active Site Of Protein Kinase Enzymes ROCK1, TNK2, GRK1 ALDH1A1 3779/4885ALPL 2276/4885CYP3A4 1134/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.