SCHEMBL4932778

SCHEMBL4932778

CCNc1cccc(COc2c(Cl)cc(CC(=O)O)cc2Cl)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 8/20 0.62
THRA P10827 6/20 0.62
MRGPRX4 Q96LA9 1/20 0.45
TP53 P04637 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ADRB2 P07550 1/20 0.41
ADRB3 P13945 1/20 0.41
PDE5A O76074 1/20 0.40
SIRT2 Q8IXJ6 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
SIRT3 Q9NTG7 1/20 0.40
SENP5 Q96HI0 1/20 0.40
SENP2 Q9HC62 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4933395 0.91 THRB (0.52) THRBTHRAMRGPRX4TP53GAA
SCHEMBL4926324 0.88 THRA (0.80) THRBTHRAMRGPRX4
SCHEMBL4360489 0.88 THRB (0.79) THRBTHRATP53GAAMAPT
SCHEMBL4929427 0.88 THRA (0.47) THRBTHRAMRGPRX4KMT2AMEN1
SCHEMBL5110110 0.86 SLC1A2 (0.51) THRBTHRAMRGPRX4GAAMAPT
SCHEMBL5111290 0.86 CLCN2 (0.52) THRBTHRAMRGPRX4KMT2AMEN1
SCHEMBL4932486 0.85 THRB (0.45) THRBTHRAMRGPRX4TP53GAA
SCHEMBL4930325 0.85 THRA (0.45) THRBTHRAMRGPRX4KMT2AADRB2
SCHEMBL4355861 0.84 THRB (0.44) THRBTHRAMRGPRX4TP53GAA
SCHEMBL4930726 0.83 THRB (0.43) THRBTHRAMRGPRX4TP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080221210-A1 Thyroid Receptor Agonists KARO BIO AB (SE) 2008-09-11 US disclosed
EP-1732533-A1 THYROID RECEPTOR AGONISTS KARO BIO AB (SE) 2006-12-20 EP disclosed
WO-2005092317-A1 THYROID RECEPTOR AGONISTS KARO BIO AB (SE) 2005-10-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080221210-A1 Thyroid Receptor Agonists TSHR, TRHR, THRA THRB 4/4885THRA 3/4885MRGPRX4 119/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.