SCHEMBL4947748

SCHEMBL4947748

O=C1CC=NC(C(F)(F)F)=C1CC(=O)c1cc(OCc2ccccc2)c(OCc2ccccc2)c([N+](=O)[O-])c1

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PTGES O14684 1/20 0.38
CTSV O60911 4/20 0.37
CTSL P07711 4/20 0.37
ABCB1 P08183 1/20 0.36
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MYC P01106 1/20 0.34
MAX P61244 1/20 0.34
POLB P06746 1/20 0.34
PIN1 Q13526 1/20 0.33
CYP19A1 P11511 1/20 0.33
MAPK1 P28482 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
KDM4E B2RXH2 1/20 0.33
PTPN2 P17706 1/20 0.33
PTPN1 P18031 1/20 0.33
PTPN6 P29350 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4942728 0.85 SMN1; SMN2 (0.37) PTGESCTSVCTSLABCB1MAPT
SCHEMBL3587958 0.77 PPIA (0.41) PTGESCTSVCTSLMAPTMEN1
SCHEMBL4948554 0.74 EIF4E (0.38) ABCB1MAPTPOLBPIN1CYP19A1
SCHEMBL1446822 0.74 PTGES (0.48) PTGESCTSVCTSLABCB1MAPT
SCHEMBL1446833 0.73 PTGES (0.41) PTGESCTSVCTSLABCB1MAPT
SCHEMBL1447206 0.73 CTSV (0.55) PTGESCTSVCTSLABCB1MAPT
SCHEMBL13257189 0.70 LMNA (0.61) PTGESCTSVCTSLABCB1MAPT
SCHEMBL4950971 0.67 NPC1 (0.51) ABCB1MEN1KMT2AKDM4E
SCHEMBL3586707 0.67 PTGES (0.42) PTGESCTSVCTSLMAPTMEN1
SCHEMBL3586711 0.67 PTGES (0.42) PTGESCTSVCTSLMAPTMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1907382-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS Portela & C.A. S.A (PT) 2008-04-09 EP disclosed
WO-2007013830-A1 NITROCATECHOL DERIVATIVES AS COMT INHIBITORS PORTELA & CA. S.A. (PT) 2007-02-01 WO disclosed