SCHEMBL4960187

SCHEMBL4960187

NC(=O)C1(Cc2ccncc2)CC1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 3/20 0.41
CYP19A1 P11511 5/20 0.40
ALDH1A1 P00352 3/20 0.39
KDM4E B2RXH2 2/20 0.39
GAA P10253 1/20 0.39
LOXL2 Q9Y4K0 2/20 0.39
CYP3A4 P08684 3/20 0.38
CYP2C9 P11712 2/20 0.38
CYP2D6 P10635 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
HIF1A Q16665 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
CYP1A2 P05177 2/20 0.38
KCNQ2 O43526 1/20 0.38
ALOX15 P16050 1/20 0.38
TSHR P16473 1/20 0.38
MPO P05164 1/20 0.37
ADORA3 P0DMS8 1/20 0.37
CYP2A6 P11509 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31682196 0.89 CYP2D6 (0.44) CYP17A1CYP19A1ALDH1A1KDM4EGAA
SCHEMBL23647399 0.85 ALDH1A1 (0.44) ALDH1A1KDM4EGAACYP3A4CYP2C9
SCHEMBL30589493 0.81 MAOA (0.50) ALDH1A1CYP2D6HIF1ASMN1; SMN2TSHR
SCHEMBL2469547 0.81 MAOA (0.50) ALDH1A1CYP2D6HIF1ASMN1; SMN2TSHR
SCHEMBL7043763 0.80 RECQL (0.51) CYP17A1CYP19A1KDM4ECYP3A4CYP2C9
SCHEMBL11296862 0.78 OPRM1 (0.49) ALDH1A1GAACYP2C9MEN1KMT2A
SCHEMBL16083425 0.78 OPRM1 (0.47) ALDH1A1GAALOXL2
SCHEMBL15897427 0.78 HSD11B1 (0.38) CYP3A4
SCHEMBL23660675 0.77 GPR119 (0.50) ALDH1A1
SCHEMBL7329139 0.76 ALDH1A1 (0.48) CYP19A1ALDH1A1KDM4EGAACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1893581-A1 SUBSTITUTED ARYLPYRAZOLES FOR USE AGAINST PARASITITES Pfizer Limited (GB) 2008-03-05 EP claimed
WO-2006134468-A1 SUBSTITUTED ARYLPYRAZOLES FOR USE AGAINST PARASITITES PFIZER LIMITED (GB) 2006-12-21 WO claimed