SCHEMBL4964684

SCHEMBL4964684

CCC(O)(CC)Cc1csc(NS(=O)(=O)c2cc(Cl)cc(OCCCN(C)C)c2)n1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.41
MEN1 O00255 5/20 0.38
ALDH1A1 P00352 2/20 0.38
POLB P06746 2/20 0.37
PKM P14618 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
KDM1A O60341 4/20 0.35
MAOA P21397 4/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.34
CACNA1B Q00975 3/20 0.34
CACNA1H O95180 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4967467 0.96 KMT2A (0.42) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4964911 0.87 KMT2A (0.44) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4963972 0.87 PKM (0.48) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4967543 0.84 KMT2A (0.42) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4965266 0.83 HSD11B1 (0.44) KMT2AALDH1A1
SCHEMBL4970500 0.82 HSD11B1 (0.44) KMT2AMEN1ALDH1A1POLBKDM4E
SCHEMBL4963612 0.81 KMT2A (0.39) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4964602 0.79 KMT2A (0.43) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4966262 0.77 KMT2A (0.40) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4965636 0.75 HSD11B1 (0.43) KMT2AMEN1ALDH1A1POLBCYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed