SCHEMBL4965636

SCHEMBL4965636

CCC(O)(CC)Cc1csc(NS(=O)(=O)c2ccc(CCCN(C)C)cc2Cl)n1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 5/20 0.43
HSD17B1 P14061 2/20 0.43
HSD17B2 P37059 2/20 0.43
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
POLB P06746 2/20 0.41
NMT1 P30419 1/20 0.35
SCN9A Q15858 3/20 0.35
CTPS1 P17812 3/20 0.35
ALDH1A1 P00352 2/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
KDM1A O60341 1/20 0.33
MAOA P21397 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4962705 0.97 HSD11B1 (0.42) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4964100 0.83 NMT1 (0.47) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4965593 0.83 NMT1 (0.44) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4963612 0.78 KMT2A (0.39) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4967543 0.78 KMT2A (0.42) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4966262 0.75 KMT2A (0.40) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4963210 0.75 TRPV4 (0.40) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4964602 0.75 KMT2A (0.43) HSD11B1HSD17B1HSD17B2KMT2AMEN1
SCHEMBL4964684 0.75 KMT2A (0.41) KMT2AMEN1POLBALDH1A1CYP2C9
SCHEMBL4963972 0.75 PKM (0.48) KMT2AMEN1POLBALDH1A1CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed