SCHEMBL4964716

SCHEMBL4964716

N#CCC1C=CN=C(N2CCN(c3ncccn3)CC2)N1c1nc2ccccc2s1.N#CCc1ccnc(N2CCN(c3cnccn3)CC2)n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SORD Q00796 2/20 0.35
DRD2 P14416 6/20 0.33
HTR1A P08908 5/20 0.33
HTR7 P34969 5/20 0.33
DRD4 P21917 4/20 0.33
DRD3 P35462 4/20 0.33
ADRA2A P08913 2/20 0.33
ADRA2C P18825 2/20 0.33
SLC6A2 P23975 2/20 0.33
ADRA1A P35348 2/20 0.33
HRH1 P35367 2/20 0.33
HTR2B P41595 2/20 0.33
SIGMAR1 Q99720 1/20 0.33
HTR2A P28223 4/20 0.33
IRAK4 Q9NWZ3 1/20 0.31
ADRA2B P18089 1/20 0.31
DRD1 P21728 1/20 0.31
ADRA1D P25100 1/20 0.31
HTR1D P28221 1/20 0.31
HTR1B P28222 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4197293 0.90 SORD (0.40) SORDDRD2HTR1AHTR7DRD4
Acetonitrile SCHEMBL6828681 0.88 SORD (0.38) SORDDRD2HTR1AHTR7DRD4
SCHEMBL4199997 0.86 HTR1A (0.42) SORDDRD2HTR1AHTR7DRD4
SCHEMBL4199975 0.77 NPC1 (0.40) SORD
SCHEMBL4197998 0.76 NPC1 (0.53)
SCHEMBL4198007 0.76 RAB9A (0.42) DRD4
SCHEMBL4195581 0.76 USP2 (0.52) DRD2HTR1AHTR7DRD4DRD3
SCHEMBL4197211 0.74 SCN4A (0.38)
SCHEMBL2878792 0.74 SORD (0.49) SORDDRD2DRD4DRD3
SCHEMBL4195517 0.73 DPP4 (0.40) SORD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904181-A2 JNK INHIBITORS FOR THE TREATMENT OF ENDOMETREOSIS LABORATOIRES SERONO S.A. (CH) 2008-04-02 EP disclosed
WO-2007011762-A2 JNK INHIBITORS FOR THE TREATMENT OF ENDOMETREOSIS LABORATOIRES SERONO S.A. (CH) 2007-01-25 WO disclosed