SCHEMBL4965409

SCHEMBL4965409

O=C1[N]c2c(C3CCNC3)cc(F)c(Cc3ccccc3)c2N1

nearest known ligand 0.40

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 2/20 0.40
GABRG2 P18507 1/20 0.40
GABRB3 P28472 1/20 0.40
HTR2C P28335 2/20 0.36
HTR2B P41595 2/20 0.36
HTR2A P28223 1/20 0.36
HTR1A P08908 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A4 P31645 1/20 0.35
SLC6A3 Q01959 1/20 0.35
JAK3 P52333 1/20 0.35
GABRB2 P47870 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4963859 0.81 GABRA1 (0.44) GABRA1GABRG2GABRB3HTR2CHTR1A
SCHEMBL4966050 0.78 GABRA1 (0.38) GABRA1GABRG2GABRB3HTR1ASLC6A2
Hydrochloric Acid SCHEMBL4966442 0.78 GABRA1 (0.38) GABRA1GABRG2GABRB3HTR1ASLC6A2
SCHEMBL4964907 0.73 PLAT (0.35)
SCHEMBL4977286 0.72 HTR6 (0.38) HTR2CHTR2BHTR2AHTR1ASLC6A2
SCHEMBL4977909 0.71 CXCR2 (0.34) HTR1ASLC6A2SLC6A4SLC6A3
SCHEMBL4965972 0.65 HTR6 (0.44) HTR2CHTR2BHTR1ASLC6A2SLC6A4
SCHEMBL11498275 0.65 SLC6A2 (0.50) GABRA1GABRG2GABRB3HTR2CHTR2B
SCHEMBL4964731 0.64 KIT (0.42) SLC6A2SLC6A4SLC6A3
Hydrochloric Acid SCHEMBL11198045 0.64 SLC6A2 (0.49) GABRA1GABRG2GABRB3HTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1904483-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. Hoffmann-Roche AG (CH) 2008-04-02 EP claimed
WO-2007006677-A1 BENZIMIDAZOLE DERIVATIVES AS 5-HT6,5-HT24 F. HOFFMANN-LA ROCHE AG (CH) 2007-01-18 WO claimed