SCHEMBL4965602

SCHEMBL4965602

CCCCC1CC(N(Cc2ccccc2)C(=O)c2ccccc2N)CCN1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
CHRM2 P08172 1/20 0.41
CHRM3 P20309 1/20 0.41
TRPM8 Q7Z2W7 2/20 0.41
OPRM1 P35372 3/20 0.41
UBE2M P61081 7/20 0.41
DCUN1D1 Q96GG9 7/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965590 0.80 DCUN1D1 (0.58) UBE2MDCUN1D1
SCHEMBL3871317 0.71 HDAC3 (0.39) CHRM2CHRM3
SCHEMBL1939688 0.69 FNTA (0.36) CHRM2CHRM3
SCHEMBL9905328 0.67 TACR1 (0.54)
SCHEMBL6274182 0.66 GNAI3 (0.41)
SCHEMBL26090906 0.66 MEN1 (0.44) KDM4ECHRM2CHRM3OPRM1
SCHEMBL6418644 0.66 TRPM8 (0.42) TRPM8UBE2MDCUN1D1
SCHEMBL3877432 0.65 DPP4 (0.37) CHRM2CHRM3
SCHEMBL5067770 0.65 DPP4 (0.35) CHRM2CHRM3
SCHEMBL21409263 0.63 CARM1 (0.43) KDM4ECHRM2CHRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1960359-A1 NOVEL N-SULFAMOYL-PIPERIDINEAMIDES FOR THE PROPHYLAXIS OR TREATMENT OF OBESITY AND RELATED CONDITIONS Solvay Pharmaceuticals GmbH (DE) 2008-08-27 EP disclosed
WO-2007065948-A1 NOVEL N-SULFAMOYL-PIPERIDINEAMIDES FOR THE PROPHYLAXIS OR TREATMENT OF OBESITY AND RELATED CONDITIONS SOLVAY PHARMACEUTICALS GMBH (DE) 2007-06-14 WO disclosed