SCHEMBL21409263

SCHEMBL21409263

CCCCC1CC(OCc2ccc(Br)cc2)CCN1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CARM1 Q86X55 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
AGTR2 P50052 2/20 0.41
EPHX2 P34913 1/20 0.38
BCHE P06276 1/20 0.35
ALDH1A1 P00352 4/20 0.34
KDM4E B2RXH2 1/20 0.34
ACHE P22303 1/20 0.34
HTR4 Q13639 1/20 0.34
COL1A1 P02452 1/20 0.34
HTT P42858 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MC4R P32245 2/20 0.34
MC3R P41968 2/20 0.34
MC1R Q01726 2/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
MGLL Q99685 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21409412 0.73 CARM1 (0.54) CARM1PRMT6AGTR2EPHX2BCHE
SCHEMBL1162325 0.73 BDKRB2 (0.43) CARM1PRMT6EPHX2ALDH1A1KDM4E
SCHEMBL21409115 0.72 CARM1 (0.48) CARM1PRMT6EPHX2BCHEALDH1A1
SCHEMBL5067770 0.69 DPP4 (0.35) ALDH1A1CHRM2CHRM1CHRM3
SCHEMBL2980458 0.69 ABCB1 (0.57) ALDH1A1MC4RMC3RMC1R
SCHEMBL18668584 0.68 S1PR1 (0.46) ALDH1A1KDM4EACHECHRM2CHRM1
SCHEMBL18668583 0.68 S1PR1 (0.46) ALDH1A1KDM4EACHECHRM2CHRM1
SCHEMBL17274394 0.68 CARM1 (0.44) CARM1PRMT6EPHX2ALDH1A1KDM4E
SCHEMBL6274182 0.68 GNAI3 (0.41) BCHE
SCHEMBL24493334 0.67 CARM1 (0.68) CARM1PRMT6EPHX2ALDH1A1HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3774804-A1 N-(3-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)PHENYL)BENZAMIDE DERIVATIVES Novartis AG (CH) 2021-02-17 EP disclosed
WO-2019186343-A1 N-(3-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)PHENYL)BENZAMIDE DERIVATIVES NOVARTIS AG (CH) 2019-10-03 WO disclosed