SCHEMBL4967478

SCHEMBL4967478

CCOCCCNCc1ccc2c(c1)CCc1cc(OC(N)=O)ccc1O2

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 8/20 0.49
KMT2A Q03164 3/20 0.46
ALDH1A1 P00352 2/20 0.46
MEN1 O00255 2/20 0.46
SMN1; SMN2 Q16637 5/20 0.43
THRB P10828 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
LMNA P02545 2/20 0.42
MAPK1 P28482 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.40
HTT P42858 2/20 0.38
HPGD P15428 2/20 0.38
RAB9A P51151 1/20 0.38
SLC2A1 P11166 1/20 0.36
NPC1 O15118 1/20 0.36
MCHR1 Q99705 1/20 0.36
MAPT P10636 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965138 0.90 MCHR1 (0.43) KDM4EKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL4965638 0.89 OPRM1 (0.41) SMN1; SMN2LMNASLC2A1
SCHEMBL4963457 0.88 SLC2A1 (0.42) LMNASLC2A1
SCHEMBL4966870 0.86 KDM4E (0.46) KDM4EKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL4966629 0.85 SLC2A1 (0.37) KDM4EKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL4965633 0.83 OPRM1 (0.45) KMT2AMEN1HTTRAB9ANPC1
SCHEMBL4966256 0.83 AURKA (0.35) KDM4EKMT2AALDH1A1MEN1SMN1; SMN2
SCHEMBL4965646 0.83 OPRM1 (0.41) KMT2AALDH1A1MEN1SMN1; SMN2LMNA
SCHEMBL4965252 0.83 OPRM1 (0.41) KDM4EKMT2AMEN1RAB9ASLC2A1
Hydrochloric Acid SCHEMBL4965277 0.82 OPRM1 (0.41) KMT2AALDH1A1MEN1SMN1; SMN2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1730140-B1 OPIOID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 2008-06-25 EP claimed