SCHEMBL4967778

SCHEMBL4967778

CCOc1cc(NC(C)=O)c(Cc2ccc(OC)cc2)cc1Br

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.54
MAPT P10636 4/20 0.54
MTNR1A P48039 1/20 0.43
MTNR1B P49286 1/20 0.43
HPGD P15428 2/20 0.42
HSD17B10 Q99714 1/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
HTT P42858 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP3A4 P08684 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
KDM4E B2RXH2 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968389 0.91 ALDH1A1 (0.45) ALDH1A1MAPTMTNR1AMTNR1BHPGD
SCHEMBL4965493 0.90 ALDH1A1 (0.46) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL4965832 0.85 FPR1 (0.42) ALDH1A1MAPTMTNR1AMTNR1BHPGD
SCHEMBL1252277 0.83 GABRA1 (0.44) ALDH1A1MAPTHPGDHSD17B10MEN1
SCHEMBL4965236 0.83 PDE4A (0.45) ALDH1A1MAPTMEN1KMT2ANPSR1
SCHEMBL4966867 0.82 ALDH1A1 (0.54) ALDH1A1MAPTHPGDMEN1KMT2A
SCHEMBL4967755 0.81 MAPT (0.44) ALDH1A1MAPTMTNR1AMTNR1BHPGD
SCHEMBL14116479 0.78 PDE4D (0.42) KMT2A
SCHEMBL4966888 0.78 PDE4D (0.42) KMT2A
SCHEMBL4966904 0.78 PDE4D (0.42) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed