SCHEMBL4965832

SCHEMBL4965832

COc1ccc(Cc2cc(Br)c(OC(C)C)cc2NC(C)=O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FPR1 P21462 2/20 0.42
ALDH1A1 P00352 6/20 0.41
SAE1 Q9UBE0 1/20 0.40
UBA2 Q9UBT2 1/20 0.40
MAPT P10636 2/20 0.40
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
LMNA P02545 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
PKM P14618 1/20 0.39
FPR2 P25090 1/20 0.39
MTNR1A P48039 2/20 0.39
MTNR1B P49286 2/20 0.39
KDM4E B2RXH2 1/20 0.39
BRPF1 P55201 1/20 0.39
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HSD17B1 P14061 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4968389 0.90 ALDH1A1 (0.45) ALDH1A1SAE1UBA2MAPTNPC1
SCHEMBL4966159 0.89 BRPF1 (0.40) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL4967778 0.85 ALDH1A1 (0.54) ALDH1A1SAE1UBA2MAPTNPC1
SCHEMBL4967755 0.83 MAPT (0.44) FPR1ALDH1A1SAE1UBA2MAPT
SCHEMBL4965236 0.82 PDE4A (0.45) ALDH1A1SAE1UBA2MAPTHSD17B1
SCHEMBL4966869 0.81 RXFP1 (0.45) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL1252277 0.80 GABRA1 (0.44) ALDH1A1MAPTNPC1RAB9ALMNA
SCHEMBL4968294 0.77 HTR2A (0.39) ALDH1A1LMNASMN1; SMN2
SCHEMBL4966904 0.77 PDE4D (0.42)
SCHEMBL4966888 0.77 PDE4D (0.42)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed
WO-2008101938-A1 GLUCOPYRANOSYL-SUBSTITUTED BENZYL-BENZONITRILE DERIVATIVES, MEDICAMENTS CONTAINING SUCH COMPOUNDS, THEIR USE AND PROCESS FOR THEIR MANUFACTURE BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2008-08-28 WO disclosed