SCHEMBL4968455

SCHEMBL4968455

Fc1cc(F)cc(C2CCNCC2)c1.Fc1ccc(C2CCNCC2)cc1F

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.49
MAOB P27338 1/20 0.49
QDPR P09417 1/20 0.49
HTR2C P28335 8/20 0.45
TNKS O95271 3/20 0.43
TNKS2 Q9H2K2 3/20 0.43
SLC18A3 Q16572 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SLC6A3 Q01959 1/20 0.42
APP P05067 2/20 0.40
HTR3A P46098 1/20 0.39
PARP1 P09874 1/20 0.38
KCNH2 Q12809 1/20 0.38
HTR6 P50406 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1765234 0.91 QDPR (0.56) KDM1AMAOBQDPRHTR2CTNKS
Hydrochloric Acid SCHEMBL1764764 0.90 QDPR (0.55) KDM1AMAOBQDPRHTR2CTNKS
SCHEMBL241200 0.86 SLC18A3 (0.50) QDPRHTR2CTNKSTNKS2SLC18A3
Hydrochloric Acid SCHEMBL1765191 0.84 HTR2C (0.48) QDPRHTR2CTNKSTNKS2SLC18A3
SCHEMBL16660426 0.81 HTR3A (0.59) KDM1AMAOBQDPRSLC6A2SLC6A4
SCHEMBL724585 0.81 HTR3A (0.59) KDM1AMAOBQDPRSLC6A2SLC6A4
SCHEMBL4968460 0.80 CCR2 (0.42) QDPRHTR2C
SCHEMBL29389392 0.78 HTR2A (0.46) KDM1AMAOBQDPRHTR2CSLC6A2
SCHEMBL808710 0.78 HTR2A (0.46) KDM1AMAOBQDPRHTR2CSLC6A2
SCHEMBL3384000 0.77 SLC18A3 (0.42) QDPRHTR2CSLC18A3SIGMAR1SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1963268-A1 DISUBSTITUTED PHENYLPIPERIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION Neurosearch Sweden AB (SE) 2008-09-03 EP disclosed
WO-2007065655-A1 DISUBSTITUTED PHENYLPIPERIDINES AS MODULATORS OF CORTICAL CATECHOLAMINERGIC NEUROTRANSMISSION NEUROSEARCH SWEDEN AB (SE) 2007-06-14 WO disclosed