SCHEMBL4973290

SCHEMBL4973290

CCC(O)(CC)c1csc(NS(=O)(=O)c2ccc3nsnc3c2)n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.45
KMT2A Q03164 6/20 0.43
MEN1 O00255 5/20 0.43
ALDH1A1 P00352 2/20 0.41
HSPD1 P10809 1/20 0.41
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPN5 P54829 1/20 0.41
HSPE1 P61604 1/20 0.41
POLB P06746 1/20 0.39
PIK3CD O00329 1/20 0.39
PIK3CA P42336 1/20 0.39
PIK3CB P42338 1/20 0.39
PIK3CG P48736 1/20 0.39
PKM P14618 1/20 0.38
KDM1A O60341 4/20 0.38
MAOA P21397 3/20 0.38
CCKBR P32239 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4965545 0.83 KMT2A (0.46) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4964613 0.83 ALDH1A1 (0.54) KMT2AMEN1ALDH1A1HSPD1PTPN2
SCHEMBL4962685 0.82 MEN1 (0.60) KMT2AMEN1ALDH1A1PKMKDM1A
SCHEMBL4965824 0.81 KMT2A (0.51) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4966790 0.81 KDM1A (0.45) KMT2AMEN1ALDH1A1KDM1AMAOA
SCHEMBL4964738 0.80 KMT2A (0.50) KMT2AMEN1ALDH1A1POLBPKM
SCHEMBL4963112 0.80 KMO (0.55) TSHRKMT2AMEN1ALDH1A1PKM
SCHEMBL4964673 0.80 KDM1A (0.53) KMT2AMEN1ALDH1A1KDM1AMAOA
SCHEMBL4965281 0.78 MEN1 (0.64) KMT2AMEN1ALDH1A1KDM1AMAOA
SCHEMBL4963200 0.78 ALDH1A1 (0.55) ALDH1A1PKMKDM1AMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP claimed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO claimed
EP-1888544-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS Takeda San Diego, Inc. (US) 2008-02-20 EP disclosed
WO-2006066109-A2 HYDROXYSTEROID DEHYDROGENASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-06-22 WO disclosed