SCHEMBL4975773

SCHEMBL4975773

Cc1ccc(-c2ccccc2)c(CCN(c2cccnc2)c2cccnc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 5/20 0.39
KCNH2 Q12809 2/20 0.39
MAPT P10636 2/20 0.38
NPC1 O15118 2/20 0.38
TP53 P04637 2/20 0.38
RAB9A P51151 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
CYP17A1 P05093 1/20 0.37
CYP2A6 P11509 2/20 0.37
KCNN4 O15554 1/20 0.36
ALDH1A1 P00352 4/20 0.36
HPGD P15428 3/20 0.36
HSD17B10 Q99714 2/20 0.36
POLB P06746 1/20 0.36
TSHR P16473 1/20 0.36
PSMB5 P28074 1/20 0.36
MAP2K4 P45985 1/20 0.36
CYP11B1 P15538 1/20 0.36
CYP11B2 P19099 1/20 0.36
PDE5A O76074 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4980305 0.85 KCNA5 (0.39) KCNA5KCNH2NPC1RAB9ACYP11B1
SCHEMBL4979253 0.85 CYP11B2 (0.46) KCNA5KCNH2CYP11B1CYP11B2PDE5A
SCHEMBL4979558 0.82 CYP11B2 (0.48) KCNA5KCNH2CYP17A1CYP11B1CYP11B2
SCHEMBL4977530 0.82 CYP11B1 (0.48) KCNA5KCNH2CYP11B1CYP11B2CYP3A4
SCHEMBL4977669 0.81 CYP11B1 (0.54) KCNA5KCNH2ALDH1A1HPGDHSD17B10
SCHEMBL4977077 0.81 CYP11B1 (0.53) MAPTNPC1RAB9ASMN1; SMN2ALDH1A1
SCHEMBL4982009 0.80 MKNK1 (0.47) KCNA5KCNH2TSHRCYP11B1CYP11B2
SCHEMBL4975675 0.80 MKNK1 (0.47) KCNA5NPC1RAB9ACYP11B1CYP11B2
SCHEMBL4974371 0.79 KCNA5 (0.50) KCNA5KCNH2MAPTTP53SMN1; SMN2
SCHEMBL4975470 0.78 KCNA5 (0.51) KCNA5KCNH2MAPTKCNN4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed