SCHEMBL4980305

SCHEMBL4980305

Clc1ccc(-c2ccccc2)c(CCN(c2cccnc2)c2cccnc2)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNA5 P22460 4/20 0.39
KCNH2 Q12809 2/20 0.39
NOS3 P29474 1/20 0.39
NOS1 P29475 1/20 0.39
NOS2 P35228 1/20 0.39
FFAR1 O14842 1/20 0.37
FFAR4 Q5NUL3 1/20 0.37
CYP11B1 P15538 2/20 0.36
CYP11B2 P19099 2/20 0.36
PDE5A O76074 2/20 0.35
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
CYP1A2 P05177 2/20 0.35
CYP2C19 P33261 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35
LMNA P02545 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
PKM P14618 1/20 0.35
GPBAR1 Q8TDU6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4979253 0.85 CYP11B2 (0.46) KCNA5KCNH2FFAR1FFAR4CYP11B1
SCHEMBL4975773 0.85 KCNA5 (0.39) KCNA5KCNH2CYP11B1CYP11B2PDE5A
SCHEMBL4979558 0.82 CYP11B2 (0.48) KCNA5KCNH2CYP11B1CYP11B2MAPK1
SCHEMBL4977530 0.82 CYP11B1 (0.48) KCNA5KCNH2CYP11B1CYP11B2CYP3A4
SCHEMBL4982009 0.80 MKNK1 (0.47) KCNA5KCNH2CYP11B1CYP11B2HTT
SCHEMBL4974371 0.79 KCNA5 (0.50) KCNA5KCNH2CYP11B1CYP11B2CYP1A2
SCHEMBL4977077 0.78 CYP11B1 (0.53) CYP11B1CYP11B2CYP2C19NPSR1LMNA
SCHEMBL4977669 0.78 CYP11B1 (0.54) KCNA5KCNH2CYP11B1CYP11B2CYP1A2
SCHEMBL4975675 0.78 MKNK1 (0.47) KCNA5CYP11B1CYP11B2LMNANPC1
SCHEMBL4975470 0.78 KCNA5 (0.51) KCNA5KCNH2CYP11B1CYP11B2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP disclosed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO disclosed