SCHEMBL4979253

SCHEMBL4979253

Fc1ccc(-c2ccccc2)c(CCN(c2cccnc2)c2cccnc2)c1

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP11B2 P19099 4/20 0.46
CYP11B1 P15538 3/20 0.46
KCNA5 P22460 6/20 0.42
KCNH2 Q12809 5/20 0.42
TDO2 P48775 1/20 0.37
FFAR1 O14842 2/20 0.37
FFAR4 Q5NUL3 2/20 0.37
RPS6KA3 P51812 1/20 0.36
GBA1 P04062 1/20 0.36
ELOVL1 Q9BW60 1/20 0.36
PDE5A O76074 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4975773 0.85 KCNA5 (0.39) CYP11B2CYP11B1KCNA5KCNH2PDE5A
SCHEMBL4980305 0.85 KCNA5 (0.39) CYP11B2CYP11B1KCNA5KCNH2FFAR1
SCHEMBL4977530 0.84 CYP11B1 (0.48) CYP11B2CYP11B1KCNA5KCNH2
SCHEMBL4979558 0.82 CYP11B2 (0.48) CYP11B2CYP11B1KCNA5KCNH2
SCHEMBL4982009 0.80 MKNK1 (0.47) CYP11B2CYP11B1KCNA5KCNH2
SCHEMBL4974371 0.79 KCNA5 (0.50) CYP11B2CYP11B1KCNA5KCNH2
SCHEMBL4977077 0.78 CYP11B1 (0.53) CYP11B2CYP11B1
SCHEMBL4977669 0.78 CYP11B1 (0.54) CYP11B2CYP11B1KCNA5KCNH2
SCHEMBL4975675 0.78 MKNK1 (0.47) CYP11B2CYP11B1KCNA5RPS6KA3
SCHEMBL4975470 0.78 KCNA5 (0.51) CYP11B2CYP11B1KCNA5KCNH2RPS6KA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1993551-A2 POTASSIUM CHANNEL INHIBITORS Merck & Co., Inc. (US) 2008-11-26 EP claimed
WO-2007089735-A2 POTASSIUM CHANNEL INHIBITORS MERCK & CO., INC. (US) 2007-08-09 WO claimed