SCHEMBL4979634

SCHEMBL4979634

O=C(O)CC1CC(=O)NC1=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB1 P05556 2/20 0.50
ITGA5 P08648 2/20 0.50
ITGB3 P05106 1/20 0.50
ITGB2 P05107 1/20 0.50
ITGAV P06756 1/20 0.50
ITGA2B P08514 1/20 0.50
ITGB5 P18084 1/20 0.50
ITGAL P20701 1/20 0.50
TSHR P16473 2/20 0.42
HTT P42858 2/20 0.42
KDM4E B2RXH2 1/20 0.42
MAP3K14 Q99558 1/20 0.40
CRBN Q96SW2 6/20 0.38
DDB1 Q16531 4/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
MEN1 O00255 1/20 0.38
APEX1 P27695 1/20 0.38
KMT2A Q03164 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
GLA P06280 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15602681 0.82 FOLH1 (0.43) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL28048806 0.82 MAP3K14 (0.39) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL11872852 0.82 GLA (0.40) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL19585667 0.80 CRBN (0.58) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL24885110 0.79 TDP1 (0.40) ITGB1ITGA5ITGB3ITGB2ITGAV
SCHEMBL28479332 0.77 MAP3K14 (0.50) MAP3K14CRBNDDB1GLAMAPT
SCHEMBL24885111 0.76 ABL1 (0.47) TSHRL3MBTL1MEN1KMT2ATDP1
SCHEMBL5779882 0.76
SCHEMBL19839455 0.76
SCHEMBL2915829 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 39 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117486998-A Dipolyethylene glycol-insulin conjugate and preparation method and application thereof 中山大学 2024-02-02 CN claimed
CN-118742317-A Liver targeting substances and uses thereof 韩美药品株式会社 2024-10-01 CN disclosed
CN-117615775-A Therapeutic uses comprising combinations of triple agonists that are all active on glucagon, GLP-1 and GIP receptors 韩美药品株式会社 2024-02-27 CN disclosed
CN-117486998-A Dipolyethylene glycol-insulin conjugate and preparation method and application thereof 中山大学 2024-02-02 CN disclosed
CN-117486998-A Dipolyethylene glycol-insulin conjugate and preparation method and application thereof 中山大学 2024-02-02 CN disclosed
CN-117462693-A XTEN conjugate compositions and methods of making the same 阿穆尼克斯运营公司 2024-01-30 CN disclosed
CN-117427179-A Chemical modifier of human urinary kallidinogenase 江苏艾迪药业股份有限公司 2024-01-23 CN disclosed
US-11834553-B2 Alkoxylation methods NEKTAR THERAPEUTICS (US) 2023-12-05 US disclosed
CN-116635055-A Pharmaceutical composition for preventing or treating lupus-related diseases comprising GIP derivative or long-acting conjugate thereof 韩美药品株式会社 2023-08-22 CN disclosed
CN-116583533-A GIP derivative, long-acting conjugate thereof and pharmaceutical composition comprising the same 韩美药品株式会社 2023-08-11 CN disclosed
US-6881396-B2 Stabilization of radiopharmaceutical compositions using hydrophilic 6-hydroxy-chromans DIATIDE, INC. (US) 2005-04-19 US disclosed
US-20040058984-A1 Stabilization of radiopharmaceutical compositions using hydrophilic thioethers and hydrophilic 6-hydroxy chromans DIATIDE LABORATORIES 2004-03-25 US disclosed
EP-1381397-A2 STABILISATION OF RADIOPHARMACEUTICAL COMPOSITIONS USING A HYDROPHILIC THIOETHER OR A HYDROPHILIC 6-HYDROXY CHROMAN Diatide, Inc. (US) 2004-01-21 EP disclosed
EP-0804252-B1 MONOAMINE, DIAMIDE, THIOL-CONTAINING METAL CHELATING AGENTS DIATIDE INC (US) 2003-08-13 EP disclosed
US-20030103895-A1 Stabilization of radiopharmaceutical compositions using hydrophilic thioethers and hydrophilic 6-hydroxy chromans CIS BIO INTERNATIONAL (FR) 2003-06-05 US disclosed
US-20030103899-A1 Stabilization of radiopharmaceutical compositions using hydrophilic 6-hydroxy-chromans CIS BIO INTERNATIONAL (FR) 2003-06-05 US disclosed
US-20030072709-A1 Stabilization of radiopharmaceutical compositions using hydrophilic thioethers CIS BIO INTERNATIONAL (FR) 2003-04-17 US disclosed
WO-2002060491-A2 STABILIZATION OF RADIOPHARMACEUTICAL COMPOSITIONS USING A HYDROPHILIC THIOETHER OR A HYDROPHILIC 6-HYDROXY CHROMAN DIATIDE, INC. (US) 2002-08-08 WO disclosed
EP-0804252-A2 MONOAMINE, DIAMIDE, THIOL-CONTAINING METAL CHELATING AGENTS DIATECH, INC. (US) 1997-11-05 EP disclosed
WO-1995033497-A1 MONOAMINE, DIAMIDE, THIOL-CONTAINING METAL CHELATING AGENTS DIATECH, INC. (US) 1995-12-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20030072709-A1 Stabilization of radiopharmaceutical compositions using hydrophilic thioethers TTPA, TTR, PHOSPHO1 ITGB1 2936/4885ITGA5 3968/4885ITGB3 2560/4885
US-20030103895-A1 Stabilization of radiopharmaceutical compositions using hydrophilic thioethers and hydrophilic 6-hydroxy chromans TSHR, SHBG, SLC18A1 ITGB1 3260/4885ITGA5 3768/4885ITGB3 2261/4885
US-20040058984-A1 Stabilization of radiopharmaceutical compositions using hydrophilic thioethers and hydrophilic 6-hydroxy chromans HTR6, SLC7A1, HTR7 ITGB1 3034/4885ITGA5 3132/4885ITGB3 2055/4885
US-11834553-B2 Alkoxylation methods ALK, ALKBH3, SLC10A1 ITGB1 4315/4885ITGA5 3110/4885ITGB3 2880/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.