Maleic Acid

Maleic Acid

SCHEMBL4981536

C=COC(=O)CC=CC(=O)O.O=C(O)/C=C\C(=O)O

nearest known ligand 0.38

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Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Maleic Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.38
GABRR1 P24046 2/20 0.38
GABRR2 P28476 2/20 0.38
BLM P54132 2/20 0.38
LMNA P02545 2/20 0.38
GABRR3 A8MPY1 1/20 0.38
APEX1 P27695 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
TP53 P04637 1/20 0.38
EGLN1 Q9GZT9 1/20 0.38
EGLN3 Q9H6Z9 1/20 0.38
HCAR2 Q8TDS4 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL211836 0.98 TSHR (0.39) TSHRGABRR1GABRR2BLMLMNA
SCHEMBL6061868 0.96 TSHR (0.38) TSHRGABRR1GABRR2BLMLMNA
Ammonia Solution, Strong SCHEMBL3280212 0.96 TSHR (0.38) TSHRGABRR1GABRR2BLMLMNA
Acrylic Acid SCHEMBL6444076 0.94 LMNA (0.40) TSHRGABRR1GABRR2BLMLMNA
Vinyl Chloride SCHEMBL259499 0.92 GABRR1 (0.35) TSHRGABRR1GABRR2BLMLMNA
Vinyl Chloride SCHEMBL6562575 0.92 GABRR1 (0.35) TSHRGABRR1GABRR2BLMLMNA
Acetic Acid SCHEMBL6563939 0.92 GABRR1 (0.35) TSHRGABRR1GABRR2BLMLMNA
Acrylic Acid SCHEMBL6562656 0.89 LMNA (0.36) TSHRGABRR1GABRR2BLMLMNA
Methacrylic Acid SCHEMBL4684697 0.87 GABRR1 (0.32) TSHRGABRR1GABRR2BLMLMNA
Acrylic Acid Methyl Ester SCHEMBL4672549 0.84 HCAR2 (0.41) TSHRGABRR1GABRR2BLMLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1280880-B1 LAUNDRY DETERGENT COMPOSITIONS CONTAINING A POLYMER PROCTER & GAMBLE (US) 2008-10-29 EP disclosed
US-6740633-B2 Polyelectrolyte complexes and a method for production thereof BASF AKTIENGESELLSCHAFT (DE) 2004-05-25 US disclosed
US-6596678-B2 Polyelectrolyte complex of cationic adducts or polymers of (poly)amines crosslinked with epihalohydrins, and a polyanionic polymer such as polysodium acrylate THE PROCTER & GAMBLE CO. 2003-07-22 US disclosed
US-20030078185-A1 Polyelectrolyte complexes and a method for production thereof BASF AKTIENGESELLSCHAFT (DE) 2003-04-24 US disclosed
EP-1280880-A2 LAUNDRY DETERGENT COMPOSITIONS CONTAINING A POLYMER THE PROCTER & GAMBLE COMPANY (US) 2003-02-05 EP disclosed
US-20010056058-A1 Laundry detergent compositions containing a polymer for fabric appearance improvement THE PROCTER & GAMBLE COMPANY 2001-12-27 US disclosed
WO-2001085891-A2 LAUNDRY DETERGENT COMPOSITIONS CONTAINING A POLYMER THE PROCTER & GAMBLE COMPANY (US) 2001-11-15 WO disclosed
US-5126411-A For coatings, films, fibers, adhesives HOECHST AG (DE) 1992-06-30 US disclosed
US-5089570-A Protective colloids HOECHST AKTIENGESELLSCHAFT (DE) 1992-02-18 US disclosed