SCHEMBL498487

SCHEMBL498487

C=CC(=O)CC(=O)C=C(c1ccc(O)c(OC)c1)c1ccc(O)c(OC)c1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
SLC22A6 Q4U2R8 1/20 0.54
SLC22A8 Q8TCC7 1/20 0.54
RAB9A P51151 1/20 0.54
HTT P42858 2/20 0.53
ALOX5 P09917 3/20 0.51
NFKB1 P19838 2/20 0.51
STAT3 P40763 2/20 0.51
NFKB2 Q00653 2/20 0.51
RELA Q04206 2/20 0.51
HSD17B2 P37059 2/20 0.50
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
TSHR P16473 2/20 0.49
HSD17B10 Q99714 2/20 0.49
CYP1A2 P05177 2/20 0.49
KDM4E B2RXH2 2/20 0.49
POLB P06746 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10771572 0.87 MEN1 (0.55) MEN1KMT2ASLC22A6SLC22A8RAB9A
SCHEMBL1672224 0.84 KDM4E (0.63) MEN1KMT2ACYP2D6TSHRKDM4E
SCHEMBL1490943 0.84 MEN1 (0.58) MEN1KMT2ASLC22A6SLC22A8RAB9A
SCHEMBL16061281 0.80 HTT (0.55) MEN1KMT2ASLC22A6SLC22A8RAB9A
SCHEMBL9579837 0.78 HTT (0.54) MEN1KMT2ASLC22A6SLC22A8RAB9A
SCHEMBL20897645 0.78 SLC22A6 (0.62) MEN1KMT2ASLC22A6SLC22A8RAB9A
SCHEMBL13733100 0.78 PKM (0.53) RAB9AKDM4EHDAC6ALDH1A1MAPT
SCHEMBL3751049 0.77 SLC22A6 (0.66) MEN1KMT2ASLC22A6SLC22A8RAB9A
SCHEMBL3731235 0.76 MEN1 (0.49) MEN1KMT2ASLC22A6SLC22A8RAB9A
Curcumin SCHEMBL15229772 0.75 APP (0.86) MEN1KMT2AHTTALOX5NFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 139 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008051474-A1 WATER SOLUBLE CURCUMIN-BASED COMPOUNDS THE UAB RESEARCH FOUNDATION (US) 2008-05-02 WO claimed
EP-1085860-B1 FORMULATIONS FOR THE TREATMENT OF GASTRO-OESOPHAGEAL REFLUX RECKITT BENCKISER HEALTHCARE (GB) 2002-10-16 EP claimed
US-20230241006-A1 CURCUMIN COMPOSITIONS FOR OSTEOARTHRITIS AND JOINT WELLNESS OMNIACTIVE HEALTH TECHNOLOGIES LIMITED (IN) 2023-08-03 US disclosed
WO-2023111967-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF THE RESPIRATORY INFECTION CAUSED BY SARS-COV-2 ALPARIS S.A. DE C.V (MX) 2023-06-22 WO disclosed
CN-115524923-A Negative photosensitive resin composition, and patterning method and application thereof 深圳市容大感光科技股份有限公司 2022-12-27 CN disclosed
US-20220387454-A1 NUTRITIONAL COMPOSITION FOR VISUAL FUNCTION OMNIACTIVE HEALTH TECHNOLOGIES LIMITED (IN) 2022-12-08 US disclosed
EP-3233068-B1 A PROCESS FOR PREPARATION OF BIOAVAILABLE WHITE CURCUMIN - A UNIQUE BLEND OF HYDROGENATED CURCUMINOIDS AUREA BIOLABS PRIVATE LTD (IN) 2021-06-16 EP disclosed
WO-2021094918-A1 NUTRITIONAL COMPOSITION FOR VISUAL FUNCTION OMNIACTIVE HEALTH TECHNOLOGIES LIMITED (IN) 2021-05-20 WO disclosed
EP-2379109-B1 COMBINATION OF PHOTODYNAMIC THERAPY AND ANTI-VEGF AGENTS IN THE TREATMENT OF UNWANTED CHOROIDAL NEOVASCULATURE BAUSCH HEALTH COMPANIES INC (CA) 2020-10-07 EP disclosed
US-10639285-B2 Process for preparation of bioavailable white curcumin—a unique blend of hydrogenated curcuminoids Aurea Biolabs Private Limited (IN) 2020-05-05 US disclosed
EP-2294186-B1 INDUCING CELL DEATH BY INHIBITING ADAPTIVE HEAT SHOCK RESPONSE INCURON INC (US) 2019-10-09 EP disclosed
WO-2001085213-A2 SUPPORTS FOR PHOTOSENSITIZER FORMULATIONS THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2001-11-15 WO disclosed
WO-2001085212-A2 DRUG DELIVERY SYSTEMS FOR PHOTODYNAMIC THERAPY THE UNIVERSITY OF BRITISH COLUMBIA (CA) 2001-11-15 WO disclosed
WO-2001035996-A2 USE OF PDT TO INHIBIT INTIMAL HYPERPLASIA QLT INC. (CA) 2001-05-25 WO disclosed
WO-2001035997-A2 USE OF LOW-DOSE PDT TO INHIBIT RESTENOSIS QLT INC. (CA) 2001-05-25 WO disclosed
EP-1085860-A1 FORMULATIONS FOR THE TREATMENT OF GASTRO-OESOPHAGEAL REFLUX RECKITT & COLMAN PRODUCTS LIMITED (GB) 2001-03-28 EP disclosed
WO-2000070949-A1 METHOD FOR USING SOLUBLE CURCUMIN TO INHIBIT PHOSPHORYLASE KINASE IN INFLAMMATORY DISEASES HENG MADALENE C Y (US) 2000-11-30 WO disclosed
WO-1999063986-A1 FORMULATIONS FOR THE TREATMENT OF GASTRO-OESOPHAGEAL REFLUX RECKITT & COLMAN PRODUCTS LIMITED (GB) 1999-12-16 WO disclosed
EP-0601882-B1 Polycarbonate resin/silicone rubber integrally molded article and method for making SHINETSU CHEMICAL CO (JP) 1998-03-11 EP disclosed
EP-0601882-A1 Polycarbonate resin/silicone rubber integrally molded article and method for making SHIN-ETSU CHEMICAL CO., LTD. (JP) 1994-06-15 EP disclosed