SCHEMBL13733100

SCHEMBL13733100

C=CC(=O)CC(=O)C=C(c1ccc(OC)cc1)c1ccc(OC)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.53
TGM2 P21980 1/20 0.49
CA1 P00915 5/20 0.49
CA2 P00918 5/20 0.49
MAPT P10636 2/20 0.49
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
GSK3B P49841 2/20 0.46
ALDH1A1 P00352 2/20 0.46
KDM4E B2RXH2 1/20 0.46
HPGD P15428 1/20 0.46
PLK1 P53350 1/20 0.46
HDAC3 O15379 1/20 0.45
HDAC4 P56524 1/20 0.45
HDAC1 Q13547 1/20 0.45
HDAC7 Q8WUI4 1/20 0.45
HDAC2 Q92769 1/20 0.45
HDAC10 Q969S8 1/20 0.45
HDAC11 Q96DB2 1/20 0.45
HDAC8 Q9BY41 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1490910 0.81 CES2 (0.52) PKMTGM2CA1CA2MAPT
SCHEMBL9176959 0.80 ALDH1A1 (0.49) CA1CA2MAPTGSK3BALDH1A1
SCHEMBL2731511 0.80 ALDH5A1 (0.52) PKMCA1CA2MAPTALDH1A1
SCHEMBL498487 0.78 MEN1 (0.54) PKMCA1CA2MAPTGSK3B
SCHEMBL2019776 0.75 CA1 (0.61) CA1CA2MAPTCES2CES1
SCHEMBL31119870 0.74 HDAC3 (0.61) PKMTGM2CA1CA2MAPT
SCHEMBL9574425 0.74 PDE4A (0.62) CA1CA2MAPTCES2CES1
SCHEMBL1672224 0.74 KDM4E (0.63) MAPTALDH1A1KDM4E
SCHEMBL546672 0.73 F3 (0.59) PKMTGM2CA1CA2MAPT
SCHEMBL3152379 0.73 HTT (0.58) PKMTGM2MAPTALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2887929-A2 COMPOUNDS FOR PREVENTING, REDUCING AND/OR ALLEVIATING ITCHY SKIN CONDITION(S) Symrise AG (DE) 2015-07-01 EP disclosed
WO-2012143576-A2 COMPOUNDS FOR PREVENTING, REDUCING AND/OR ALLEVIATING ITCHY SKIN CONDITION(S) SYMRISE AG (DE) 2012-10-26 WO disclosed