SCHEMBL4992669

SCHEMBL4992669

Cc1ccc(CS(=O)(=O)N2CCc3cnc(N)nc3C2)cc1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 1/20 0.43
PDGFRB P09619 5/20 0.41
KDR P35968 5/20 0.41
CNR2 P34972 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.38
KMT2A Q03164 2/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
MEN1 O00255 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
GRM5 P41594 1/20 0.36
HTR2C P28335 1/20 0.36
HTR2B P41595 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4992668 0.86 MAPK1 (0.40) MAPK1PDGFRBKDRCNR2L3MBTL1
SCHEMBL5142651 0.77 CNR2 (0.37) CNR2L3MBTL1KMT2ANPC1RAB9A
SCHEMBL3530577 0.71 MAPT (0.48) MAPK1PDGFRBKDRKMT2ANPC1
SCHEMBL5142650 0.70 CNR2 (0.38) CNR2KMT2ANPC1RAB9AMEN1
SCHEMBL2249696 0.68 PDGFRB (0.47) PDGFRBKDRKMT2ANPC1RAB9A
SCHEMBL30539315 0.66 KMT2A (0.59) L3MBTL1KMT2AMEN1POLB
SCHEMBL7821841 0.66 KMT2A (0.59) L3MBTL1KMT2AMEN1POLB
SCHEMBL19151139 0.65 ALDH1A1 (0.48) KMT2AMEN1LMNAPOLB
SCHEMBL4982513 0.65 L3MBTL1 (0.46) CNR2L3MBTL1
SCHEMBL4988108 0.65 GPR183 (0.36) CNR2KMT2AMEN1LMNAGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080039478-A1 Bicycloheteroaryl Compounds as P2X7 Modulators and Uses Thereof RENOVIS, INC. 2008-02-14 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080039478-A1 Bicycloheteroaryl Compounds as P2X7 Modulators and Uses Thereof P2RX7, P2RX3, P2RX2 MAPK1 546/4885PDGFRB 1740/4885KDR 3574/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.