SCHEMBL5010443

SCHEMBL5010443

O=C(O)c1cc(NC(=O)c2ccc(Cl)cc2Cl)[nH]n1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 2/20 0.56
PPARA Q07869 1/20 0.56
MEN1 O00255 3/20 0.54
KMT2A Q03164 3/20 0.54
L3MBTL1 Q9Y468 2/20 0.54
ALPL P05186 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.54
TSHR P16473 1/20 0.54
CASP1 P29466 1/20 0.54
JAK2 O60674 1/20 0.52
JAK1 P23458 1/20 0.52
TYK2 P29597 1/20 0.52
PYGL P06737 3/20 0.51
LMNA P02545 1/20 0.50
NPC1 O15118 5/20 0.49
RAB9A P51151 5/20 0.49
MAPT P10636 3/20 0.49
KDM4E B2RXH2 1/20 0.49
HDAC1 Q13547 1/20 0.48
HDAC8 Q9BY41 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3798963 0.84 BDKRB1 (0.51) KMT2ASMN1; SMN2JAK2JAK1TYK2
SCHEMBL5010776 0.82 GAA (0.56) PPARGMEN1KMT2AL3MBTL1ALPL
SCHEMBL3822963 0.81 PYGL (0.50) MEN1KMT2ASMN1; SMN2PYGLLMNA
SCHEMBL5013483 0.80 GPR27 (0.44) MEN1KMT2AALPLPYGLNPC1
Benzamide SCHEMBL27706773 0.78 PYGL (0.45) KMT2APYGLNPC1RAB9AHPGD
Benzamide SCHEMBL27727800 0.78 CYP11B2 (0.45) PPARGPPARAMEN1KMT2ANPC1
SCHEMBL3794816 0.78 NPC1 (0.56) MEN1KMT2ASMN1; SMN2TSHRJAK2
SCHEMBL5867536 0.77 MEN1 (0.51) PPARGPPARAMEN1KMT2AL3MBTL1
SCHEMBL1308769 0.76 PPARG (0.69) PPARGPPARAMEN1KMT2ASMN1; SMN2
SCHEMBL14587853 0.75 GAA (0.70) MEN1KMT2ASMN1; SMN2TSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1884513-A1 PYRAZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES COMPRISING THE SAME Japan Tobacco, Inc. (JP) 2008-02-06 EP claimed
US-20070032529-A1 Pyrazole compounds and their use as antidiabetes agents JAPAN TOBACCO INC. (JP) 2007-02-08 US claimed
EP-1884513-A1 PYRAZOLE COMPOUND AND THERAPEUTIC AGENT FOR DIABETES COMPRISING THE SAME Japan Tobacco, Inc. (JP) 2008-02-06 EP disclosed
US-20070032529-A1 Pyrazole compounds and their use as antidiabetes agents JAPAN TOBACCO INC. (JP) 2007-02-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070032529-A1 Pyrazole compounds and their use as antidiabetes agents PYGL, GYS2, AGL PPARG 706/4885PPARA 1127/4885MEN1 4075/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.