SCHEMBL5012256

SCHEMBL5012256

Cc1ccc(CNC(=O)ON2C(c3ccc(Cl)cc3)=NOC23CCCCC3)cc1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TP53 P04637 3/20 0.46
LMNA P02545 2/20 0.46
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
THRB P10828 2/20 0.41
GLA P06280 1/20 0.41
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 2/20 0.39
MAPK1 P28482 1/20 0.38
CHRM1 P11229 1/20 0.38
HTR2A P28223 1/20 0.38
MCHR1 Q99705 1/20 0.38
SSTR3 P32745 1/20 0.38
POLB P06746 1/20 0.37
TSHR P16473 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5014558 0.89 LMNA (0.38) TP53LMNANPC1RAB9AMEN1
SCHEMBL5012836 0.77 ALDH1A1 (0.49) TP53LMNANPC1RAB9ATHRB
SCHEMBL5010991 0.74 TRPV1 (0.41) TP53LMNANPC1RAB9ATHRB
SCHEMBL16175419 0.73 KMT2A (0.47) TP53LMNANPC1RAB9AGLA
SCHEMBL5048772 0.72 P2RY12 (0.41) TP53
SCHEMBL16175692 0.67 KMT2A (0.50) TP53GLAMEN1KMT2AALDH1A1
SCHEMBL5012907 0.65 TSHR (0.46) LMNATHRBALDH1A1CHRM1TSHR
SCHEMBL5123358 0.65 KMT2A (0.49) TP53LMNANPC1RAB9AGLA
SCHEMBL16175732 0.64 KMT2A (0.49) LMNAMEN1KMT2AALDH1A1MAPT
SCHEMBL2096445 0.63 SMN1; SMN2 (0.64) LMNANPC1RAB9ATHRBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1888596-A1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS Grünenthal GmbH (DE) 2008-02-20 EP claimed
WO-2006122770-A1 SUBSTITUTED SPIRO COMPOUNDS AND THEIR USE FOR PRODUCING PAIN-RELIEF MEDICAMENTS Grünenthal GmbH (DE) 2006-11-23 WO claimed