SCHEMBL5024474

SCHEMBL5024474

OCCOc1ccc(C#CC(O)c2ccccc2)cc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
RECQL P46063 1/20 0.53
GAA P10253 1/20 0.46
APP P05067 6/20 0.43
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42
CHRNA3 P32297 1/20 0.42
CHRNA7 P36544 1/20 0.42
CHRNA4 P43681 1/20 0.42
TSHR P16473 1/20 0.41
FFAR1 O14842 1/20 0.41
LTA4H P09960 1/20 0.40
BRD4 O60885 1/20 0.39
CREBBP Q92793 1/20 0.39
PKM P14618 1/20 0.39
NR1I2 O75469 1/20 0.38
CYP19A1 P11511 1/20 0.38
CACNA2D1 P54289 1/20 0.38
CACNB2 Q08289 1/20 0.38
CACNA1C Q13936 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5172544 0.85 APP (0.41) ALDH1A1RECQLAPPNR1I2
SCHEMBL1819985 0.85 MCHR1 (0.48) ALDH1A1RECQLAPPTSHRNR1I2
SCHEMBL22122710 0.81 LTA4H (0.50) CHRNB2CHRNB4CHRNA3CHRNA7CHRNA4
SCHEMBL2685285 0.80 APP (0.49) ALDH1A1APPLTA4HCACNA2D1CACNB2
SCHEMBL23572596 0.80 APP (0.49) ALDH1A1APPLTA4HCACNA2D1CACNB2
SCHEMBL2519799 0.78 TSHR (0.52) ALDH1A1APPTSHRFFAR1PKM
SCHEMBL2801832 0.78 TSHR (0.52) ALDH1A1APPTSHRFFAR1PKM
SCHEMBL1819239 0.77 MAPT (0.41) ALDH1A1GAAMAPK1
SCHEMBL9553407 0.76 BCHE (0.50) ALDH1A1
SCHEMBL12711671 0.76 APP (0.65) ALDH1A1RECQLGAAAPPFFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1872173-A1 PHOTOCHROMIC MATERIALS HAVING EXTENDED PI-CONJUGATED SYSTEMS AND COMPOSITIONS AND ARTICLES INCLUDING THE SAME TRANSITIONS OPTICAL, INC. (US) 2008-01-02 EP disclosed
EP-1869140-A1 OPHTHALMIC DEVICES COMPRISING PHOTOCHROMIC MATERIALS HAVING EXTENDED PI-CONJUGATED SYSTEMS Johnson and Johnson Vision Care, Inc. (US) 2007-12-26 EP disclosed
WO-2006110513-A1 OPHTHALMIC DEVICES COMPRISING PHOTOCHROMIC MATERIALS HAVING EXTENDED PI-CONJUGATED SYSTEMS JOHNSON & JOHNSON VISION CARE, INC. (US) 2006-10-19 WO disclosed
WO-2006110221-A1 PHOTOCHROMIC MATERIALS HAVING EXTENDED PI-CONJUGATED SYSTEMS AND COMPOSITIONS AND ARTICLES INCLUDING THE SAME TRANSITIONS OPTICAL, INC. (US) 2006-10-19 WO disclosed