SCHEMBL5029975

SCHEMBL5029975

C=C(C(=O)O)c1cc2ccccc2n1S(=O)(=O)c1ccccc1Br

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.44
ALDH1A1 P00352 3/20 0.43
LMNA P02545 1/20 0.43
MAPT P10636 1/20 0.43
ACLY P53396 1/20 0.41
HDAC3 O15379 2/20 0.40
HDAC4 P56524 2/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC7 Q8WUI4 2/20 0.40
HDAC2 Q92769 2/20 0.40
HDAC10 Q969S8 2/20 0.40
HDAC11 Q96DB2 2/20 0.40
HDAC8 Q9BY41 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
HDAC9 Q9UKV0 2/20 0.40
HDAC5 Q9UQL6 2/20 0.40
NOD2 Q9HC29 4/20 0.40
NOD1 Q9Y239 4/20 0.40
TSHR P16473 1/20 0.40
DAO P14920 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3561901 0.76 ACLY (0.46) ACLYTSHRCA12CA2CA9
SCHEMBL6829943 0.75 HTR6 (0.46) ALDH1A1ACLYTSHRALOX5
SCHEMBL3563939 0.75 ACLY (0.62) ACLYCA12CA2CA9
SCHEMBL15657021 0.69 MCL1 (0.70) ALDH1A1MAPTTSHRDAOMCL1
SCHEMBL29945775 0.69 MCL1 (0.70) ALDH1A1MAPTTSHRDAOMCL1
SCHEMBL14399008 0.69 CCR2 (0.55) CCR2ALDH1A1LMNAMAPTACLY
SCHEMBL4121234 0.68 CCR2 (0.72) CCR2ALDH1A1LMNAMAPTHDAC3
SCHEMBL6864420 0.68 ALDH1A1 (0.73) CCR2ALDH1A1LMNAMAPTHDAC3
SCHEMBL31599460 0.68 CCR2 (0.72) CCR2ALDH1A1LMNAMAPTHDAC3
Hydrochloric Acid SCHEMBL4119324 0.67 CCR2 (0.71) CCR2ALDH1A1LMNAMAPTHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1990335-A1 17 BETA HSD TYPE 5 INHIBITOR Astellas Pharma Inc. (JP) 2008-11-12 EP disclosed