SCHEMBL5031121

SCHEMBL5031121

NC(=O)C1(C(=O)N2CCOCC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.47
MAPK1 P28482 1/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
MEN1 O00255 1/20 0.41
TP53 P04637 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 2/20 0.41
KDM4E B2RXH2 2/20 0.39
MMP1 P03956 1/20 0.39
MMP3 P08254 1/20 0.39
MMP8 P22894 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.38
LMNA P02545 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3551350 0.81 HSD11B1 (0.41) SMN1; SMN2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL5027626 0.81 HSD11B1 (0.36) SMN1; SMN2MEN1TP53KMT2AALDH1A1
SCHEMBL5031157 0.79 HSD11B1 (0.42) GAASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL30635290 0.76 HSD11B1 (0.46) MEN1KMT2ALMNA
SCHEMBL22720076 0.76 GAA (0.47) GAAMAPK1SMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL5031123 0.75 GAA (0.50) GAAMAPK1SMN1; SMN2CA12CA1
SCHEMBL28543459 0.73 MEN1 (0.43) GAASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL7176021 0.73 MEN1 (0.43) GAASMN1; SMN2MEN1KMT2AALDH1A1
SCHEMBL24680905 0.73 GAA (0.45) GAAMAPK1SMN1; SMN2ALDH1A1L3MBTL1
SCHEMBL4562587 0.72 RBP4 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7429609-B2 Pyrazole compound and medicinal composition containing the same EISAI R & D MANAGEMENT CO., LTD. (JP) 2008-09-30 US disclosed
EP-1510516-A1 PYRAZOLE COMPOUND AND MEDICINAL COMPOSITION CONTAINING THE SAME Eisai Co., Ltd. (JP) 2005-03-02 EP disclosed