SCHEMBL5031380

SCHEMBL5031380

CCCCNc1ccc([N+](=O)[O-])cc1C#C[Si](C)(C)C

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.50
MAPT P10636 6/20 0.47
SMN1; SMN2 Q16637 3/20 0.47
LMNA P02545 1/20 0.47
MAPK1 P28482 1/20 0.47
CCNT1 O60563 1/20 0.47
CDK9 P50750 1/20 0.47
RECQL P46063 1/20 0.47
POLB P06746 4/20 0.44
HCAR3 P49019 2/20 0.44
PKM P14618 2/20 0.44
ALDH1A1 P00352 3/20 0.44
KAT2B Q92831 1/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.42
MEN1 O00255 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP19A1 P11511 2/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9373869 0.79 RECQL (0.66) RIPK1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL1465733 0.77 MEN1 (0.41) MAPTSMN1; SMN2LMNARECQLPOLB
SCHEMBL28632584 0.77 RECQL (0.47) RIPK1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL14294847 0.76 MAPT (0.69) RIPK1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL9507998 0.75 MAPT (0.54) RIPK1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL10489384 0.73 KAT2B (0.74) RIPK1MAPTSMN1; SMN2LMNAMAPK1
SCHEMBL5718688 0.73 ALDH1A1 (0.50) MAPTSMN1; SMN2ALDH1A1MEN1KMT2A
SCHEMBL12742256 0.73 ALDH1A1 (0.53) MAPTSMN1; SMN2LMNAPOLBALDH1A1
SCHEMBL27510433 0.73 HTT (0.57) MAPTSMN1; SMN2LMNAMAPK1PKM
SCHEMBL29306545 0.72 HCAR3 (0.67) RIPK1MAPTSMN1; SMN2LMNAMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007756-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS Vertex Pharmceuticals Incorporated (US) 2008-12-31 EP disclosed
WO-2007117715-A2 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2007-10-18 WO disclosed