SCHEMBL5035231

SCHEMBL5035231

Cc1ccc(S(=O)(=O)NC(C)(C)CO)cc1NC(=O)Oc1cnn2c(C3CC3)cc(-c3ccc(C(F)(F)F)cc3)nc12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF18A Q8NI77 1/20 0.35
ALDH1A1 P00352 2/20 0.34
KMT2A Q03164 2/20 0.34
HPGD P15428 1/20 0.34
KDM4E B2RXH2 3/20 0.33
CA12 O43570 1/20 0.33
CA9 Q16790 1/20 0.33
PLAT P00750 3/20 0.33
GAA P10253 2/20 0.32
MAPT P10636 1/20 0.32
GPR119 Q8TDV5 2/20 0.32
RECQL P46063 1/20 0.32
TP53 P04637 1/20 0.32
POLB P06746 1/20 0.32
TRPA1 O75762 1/20 0.31
TSHR P16473 1/20 0.31
CASP1 P29466 1/20 0.31
HTT P42858 1/20 0.31
CASP7 P55210 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5032617 0.93 TP53 (0.36) KIF18AALDH1A1KMT2AKDM4ECA12
SCHEMBL5034987 0.90 KDM4E (0.41) KIF18AALDH1A1KMT2AHPGDKDM4E
SCHEMBL5032665 0.89 KIF18A (0.46) KIF18AKMT2AKDM4EHTT
SCHEMBL5045719 0.89 POLB (0.44) KIF18AALDH1A1KMT2AKDM4EPLAT
SCHEMBL5032676 0.88 ALDH1A1 (0.45) KIF18AALDH1A1KMT2AKDM4EMAPT
SCHEMBL5041458 0.82 ALDH1A1 (0.40) KIF18AALDH1A1KMT2AHPGDKDM4E
SCHEMBL5032572 0.81 KIF18A (0.45) KIF18AKMT2AKDM4EHTT
SCHEMBL5041408 0.81 KIF18A (0.45) KIF18AKMT2AKDM4EHTT
SCHEMBL5045196 0.81 POLB (0.49) KIF18AALDH1A1KMT2AKDM4EPLAT
SCHEMBL5034997 0.81 KDM4E (0.41) KIF18AALDH1A1KMT2AHPGDKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed