SCHEMBL5033170

SCHEMBL5033170

CC(=O)c1cccc(OCC2CC2)c1OC(F)F

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE4D Q08499 12/20 0.47
PDE4B Q07343 11/20 0.47
PDE4A P27815 8/20 0.47
PDE4C Q08493 8/20 0.47
ABCB11 O95342 1/20 0.39
FAAH O00519 1/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ABCB1 P08183 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6456302 0.88 PDE4B (0.47) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL4429839 0.87 PDE4B (0.45) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL18374066 0.80 RIPK1 (0.42) PDE4DPDE4BPDE4APDE4CFAAH
SCHEMBL20207588 0.78 RIPK1 (0.43) PDE4DPDE4BPDE4APDE4CFAAH
SCHEMBL30735868 0.77 PDE4B (0.42) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL4594035 0.77 PDE4B (0.45) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL2518447 0.76 PDE4D (0.66) PDE4DPDE4BPDE4APDE4CABCB11
SCHEMBL5115860 0.75 CXCR5 (0.43) PDE4D
SCHEMBL2658234 0.75 FAAH (0.47) FAAHCNR1CNR2
SCHEMBL20207066 0.75 RIPK1 (0.40) PDE4DPDE4BPDE4APDE4CFAAH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008117943-A1 7-(3',4'-DIALKOXYPHENYL)-[1,2,4]-TRIAZOLO[1,5-A]PYRIMIDINE COMPOUNDS, PROCESS FOR PREPARING THEREOF, AND PHARMACEUTICAL COMPOSITION FOR TREATING OR PREVENTING ASTHMA, CHRONIC OBSTRUCTIVE PULMONARY DISEASE, ARTHRITIS, ATOPIC DERMATITIS, TUMOR AND DEGENERATIVE BRAIN DISEASES COMPRISING THE SAME KOREA RESEARCH INSTITUTE OF CHEMICAL TECHNOLOGY (KR) 2008-10-02 WO disclosed