SCHEMBL5035258

SCHEMBL5035258

CC(C)(CO)NS(=O)(=O)c1ccc(Cl)c(C(N)=O)c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
KDM4E B2RXH2 1/20 0.51
HTT P42858 1/20 0.42
THRB P10828 1/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 1/20 0.40
PLG P00747 1/20 0.40
PLAU P00749 1/20 0.40
PLAT P00750 1/20 0.40
TSHR P16473 2/20 0.40
POLB P06746 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
KIF18A Q8NI77 1/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
CA3 P07451 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5035106 0.85 MAPK1 (0.53) ALDH1A1L3MBTL1KDM4ELMNAPOLB
SCHEMBL5032646 0.82 KDM4E (0.54) ALDH1A1L3MBTL1KDM4ETHRBLMNA
SCHEMBL5035886 0.76 THRB (0.64) ALDH1A1L3MBTL1KDM4ETHRB
SCHEMBL5032668 0.76 ALDH1A1 (0.50) ALDH1A1L3MBTL1KDM4ELMNANPC1
SCHEMBL30079307 0.75 TSHR (0.63) ALDH1A1L3MBTL1KDM4ETSHRSMN1; SMN2
SCHEMBL13684651 0.74 PKM (0.46) ALDH1A1KDM4ETHRBLMNANPC1
SCHEMBL1940129 0.74 KDM4E (0.37) ALDH1A1L3MBTL1KDM4EPOLBCA12
SCHEMBL13545096 0.73 SMN1; SMN2 (0.47) ALDH1A1KDM4ETHRBLMNANPC1
SCHEMBL3524423 0.73 LMNA (0.62) ALDH1A1KDM4EHTTLMNANPC1
SCHEMBL5034910 0.72 KDM4E (0.56) ALDH1A1L3MBTL1KDM4EHTTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP claimed
EP-1761541-B1 PYRRAZOLO-PYRIMIDINE DERIVATIVES HOFFMANN LA ROCHE (CH) 2008-01-09 EP disclosed