SCHEMBL5044218

SCHEMBL5044218

CCCCCCCCCCCCNC(=O)c1ccc(CC([NH])c2ccc(OC(F)(F)F)cc2)c(Br)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MLYCD O95822 1/20 0.47
HDAC3 O15379 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC2 Q92769 1/20 0.44
TRPV1 Q8NER1 7/20 0.43
PDK1 Q15118 1/20 0.42
PDK2 Q15119 1/20 0.42
PDK3 Q15120 1/20 0.42
PDK4 Q16654 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.40
NAMPT P43490 1/20 0.40
EPHX2 P34913 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
MCHR1 Q99705 1/20 0.39
NCEH1 Q6PIU2 1/20 0.39
CA2 P00918 1/20 0.39
KDM4E B2RXH2 2/20 0.39
ALDH1A1 P00352 2/20 0.39
HPGD P15428 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5044228 0.90 NAMPT (0.46) MLYCDHDAC3HDAC1HDAC2TRPV1
SCHEMBL5048870 0.88 MLYCD (0.52) MLYCDHDAC3HDAC1PDK1PDK2
SCHEMBL6023237 0.87 EPHX2 (0.49) HDAC3HDAC1HDAC2TRPV1NAMPT
SCHEMBL5045572 0.82 ALDH1A1 (0.49) MLYCDHDAC3HDAC1HDAC2PDK1
SCHEMBL5044219 0.81 MLYCD (0.48) MLYCDHDAC3HDAC1HDAC2TRPV1
SCHEMBL6022083 0.81 TRPV1 (0.48) MLYCDHDAC3HDAC1HDAC2TRPV1
SCHEMBL24119885 0.79 MLYCD (0.68) MLYCDHDAC3HDAC1HDAC2TRPV1
SCHEMBL1851709 0.77 GCGR (0.48) MLYCDHDAC3HDAC1HDAC2TRPV1
SCHEMBL5044895 0.76 EPHX2 (0.48) HDAC3HDAC1HDAC2TRPV1EPHX2
SCHEMBL5044232 0.76 MAPK14 (0.49) MLYCDHDAC3HDAC1TRPV1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1732534-B1 USE OF METHYLENE AMIDE DERIVATIVES IN CARDIOVASCULAR DISORDERS SERONO LAB (CH) 2008-07-23 EP claimed