SCHEMBL5046060

SCHEMBL5046060

COc1ccc(Cn2c(-c3csc(-c4ccc(OC)cc4)n3)cc(OC(=O)NCC(C)C)c2C)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLKB1 P03952 1/20 0.43
KDM4E B2RXH2 4/20 0.42
RAB9A P51151 4/20 0.42
ALDH1A1 P00352 4/20 0.42
NPC1 O15118 3/20 0.42
SMN1; SMN2 Q16637 3/20 0.42
EIF4E P06730 1/20 0.42
MAPT P10636 4/20 0.41
POLB P06746 1/20 0.41
ATM Q13315 1/20 0.41
HPGD P15428 2/20 0.40
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPK1 P28482 1/20 0.39
CYP1A1 P04798 1/20 0.39
CYP1B1 Q16678 1/20 0.39
THRB P10828 1/20 0.39
CDC25A P30304 1/20 0.39
CDC25B P30305 1/20 0.39
CDC25C P30307 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5039574 0.90 ALDH1A1 (0.42) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5039689 0.88 MAPT (0.43) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5048718 0.87 EIF4E (0.41) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5048642 0.86 CDC25A (0.44) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5043669 0.86 KLKB1 (0.54) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5044045 0.85 THRB (0.45) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5133210 0.85 CDC25A (0.43) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5049186 0.84 NPC1 (0.41) KLKB1KDM4ERAB9AALDH1A1NPC1
SCHEMBL5046059 0.83 EIF4E (0.46) KLKB1EIF4EMAPTTP53THRB
SCHEMBL5046039 0.83 CYP3A4 (0.41) KLKB1KDM4ERAB9AALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1583762-B1 PYRROLYL-THIAZOLES AND THEIR USE AS CB 1 RECEPTOR INVERSE AGONISTS HOFFMANN LA ROCHE (CH) 2008-07-09 EP claimed