SCHEMBL5050796

SCHEMBL5050796

CCCc1nc(NC(=O)c2ccc(Cl)cc2)c(C(=O)O)n1CC(C)C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
GAA P10253 2/20 0.41
KDM4E B2RXH2 2/20 0.41
POLB P06746 1/20 0.41
CTDSP1 Q9GZU7 1/20 0.41
HPGD P15428 2/20 0.40
HTT P42858 2/20 0.40
LMNA P02545 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
MAPT P10636 1/20 0.40
CRHBP P24387 1/20 0.40
CRHR2 Q13324 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
PTGDR2 Q9Y5Y4 1/20 0.40
MCHR1 Q99705 1/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
TP53 P04637 1/20 0.39
TMIGD3 P0DMS9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4890821 0.86 ALDH1A1 (0.37) ALDH1A1GAAKDM4EPOLBCTDSP1
SCHEMBL4893882 0.80 CNR2 (0.42) ALDH1A1GAAKDM4EHPGDHTT
SCHEMBL4883267 0.67 CYP19A1 (0.47) ALDH1A1GAAHTTMEN1KMT2A
SCHEMBL11839455 0.66 RXFP1 (0.67) ALDH1A1KDM4ELMNAMEN1KMT2A
SCHEMBL4890027 0.65 ADORA3 (0.43) ALDH1A1HPGDHTTLMNAMAPT
SCHEMBL28421136 0.64 AGTR1 (0.62) AGTR1AGTR2
SCHEMBL4576546 0.64 PTGS2 (0.49) ALDH1A1GAAHPGDHTTLMNA
SCHEMBL4789019 0.62 SMN1; SMN2 (0.41) ALDH1A1KDM4EMEN1KMT2AMAPT
SCHEMBL6168957 0.62 AGTR1 (0.69) GAANPC1RAB9AAGTR1AGTR2
SCHEMBL8408236 0.62 KDM4E (0.74) ALDH1A1GAAKDM4EPOLBCTDSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1968946-A1 IMIDAZOLES AS GABA-B RECEPTOR MODULATORS AstraZeneca AB (SE) 2008-09-17 EP disclosed
WO-2007073299-A1 IMIDAZOLES AS GABA-B RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2007-06-28 WO disclosed